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Found 226 with Last Name = 'chemtob' and Initial = 's'
TargetEstrogen receptor [D538G](Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  6.08nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)
Affinity DataIC50:  6.08nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(MOUSE)
Mcgill University Health Center Research Institute

Curated by ChEMBL
LigandPNGBDBM50355549(CHEMBL1910324)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at FP receptor in mouse myometrial strip assessed as inhibition of PGF-2alpha-induced contractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Mcgill University Health Center Research Institute

Curated by ChEMBL
LigandPNGBDBM50355549(CHEMBL1910324)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at FP receptor in bovine myometrial strip assessed as inhibition of PGF-2alpha-induced contractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Ovis aries)
Mcgill University Health Center Research Institute

Curated by ChEMBL
LigandPNGBDBM50355549(CHEMBL1910324)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at FP receptor in sheep myometrial strip assessed as inhibition of PGF-2alpha-induced contractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  15.9nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394979(CHEMBL18872)
Affinity DataIC50:  62.9nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581255(CHEMBL4531645)
Affinity DataIC50:  100nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581250(CHEMBL4455562)
Affinity DataIC50:  240nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395006(CHEMBL2163473)
Affinity DataIC50:  465nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor [D538G](Homo sapiens (Human))
Valorisation-Recherche, Limited Partnership

US Patent
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50:  568nMAssay Description:GHS-R1a radioreceptor assay using LLCPK-1 membranes overexpressing GSH-R1a and radioiodinated (1-28) rat ghrelin as tracer.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395024(CHEMBL2163444 | US9708370, CP-2A(v))
Affinity DataIC50:  568nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581260(CHEMBL4528721)
Affinity DataIC50:  670nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394997(CHEMBL2163482 | US9708370, DBG-253-6)
Affinity DataIC50:  723nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395005(CHEMBL2163474)
Affinity DataIC50:  729nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395009(CHEMBL2163470)
Affinity DataIC50:  750nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394996(CHEMBL2163348 | US9708370, DBG-253-7)
Affinity DataIC50:  771nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395003(CHEMBL2163476 | US9708370, DBG-188p)
Affinity DataIC50:  808nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581254(CHEMBL4471086)
Affinity DataIC50:  890nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395009(CHEMBL2163470)
Affinity DataIC50:  1.11E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394983(CHEMBL2163466)
Affinity DataIC50:  1.17E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50:  1.34E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394999(CHEMBL2163480 | US9708370, DBG-253-3)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50:  1.34E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395004(CHEMBL2163475)
Affinity DataIC50:  1.64E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50242203(CHEMBL4078128)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395007(CHEMBL2163472)
Affinity DataIC50:  1.80E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM263222(US9708370, DBG-175p)
Affinity DataIC50:  1.80E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50049479((S)-6-Amino-2-{(R)-2-[(S)-2-{(S)-2-[(R)-2-[(S)-2-a...)
Affinity DataIC50:  1.82E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581259(CHEMBL5080816)
Affinity DataIC50:  1.86E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50394994(CHEMBL2163484 | US9708370, DBG-178p)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of photoactivatable [125I]-Tyr-Bpa-Ala-hexarelin binding to CD36 in Sprague-Dawley rat heart membranes after 60 mins by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  2.08E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581261(CHEMBL5092625)
Affinity DataIC50:  2.26E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395001(CHEMBL2163478 | US9708370, DBG-253-1)
Affinity DataIC50:  2.77E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50:  2.89E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395002(CHEMBL2163477 | US9708370, DBG-201-A)
Affinity DataIC50:  2.89E+3nMAssay Description:Displacement of photoactivatable [125I]-Tyr-Bpa-Ala-Hexarelin from CD36 in Sprague-Dawley rat cardiac membranes incubated for 60 mins by densitometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM263256(US9708370, 67 ZS555-F40 | US9708370, ZS555-F40)
Affinity DataIC50:  2.95E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails US Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  2.97E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581258(CHEMBL5094226)
Affinity DataIC50:  3.06E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394995(CHEMBL2163483 | US9708370, DBG-253-8)
Affinity DataIC50:  3.25E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50370294(Examorelin | HEXARELIN | US9708370, Hexareline)
Affinity DataIC50:  3.33E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50242204(CHEMBL4086017)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394985(CHEMBL2163464)
Affinity DataIC50:  3.61E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50395019(CHEMBL2163449 | US9708370, CP-2B(v))
Affinity DataIC50:  3.68E+3nMpH: 7.3Assay Description:Competition experiments were performed by incubating 50 μg of LLC-PK1 membranes expressing human GHS-R1a with 15 fmol of 125I-Ghrelin and increa...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394998(CHEMBL2163481 | US9708370, DBG-253-5)
Affinity DataIC50:  3.74E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394986(CHEMBL2163463)
Affinity DataIC50:  3.86E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50394982(CHEMBL2163467)
Affinity DataIC50:  4.55E+3nMAssay Description:Displacement of [125I]ghrelin expressed in in LLC-PK1 cells incubated for 1 hr by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet glycoprotein 4(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50581256(CHEMBL5087491)
Affinity DataIC50:  4.75E+3nMAssay Description:Displacement of [125I]-Tyr-Bpa-Ala-hexarelin from rat CD36 receptor in heart tissue membrane incubated for 60 mins by competitive receptor binding as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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