Affinity DataKi: 0nMAssay Description:Binding affinity to human D2 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition of Candida albicans ATCC 38247 inositol phosphorylceramide synthase preincubated for 30 minsMore data for this Ligand-Target Pair
TargetInositol phosphorylceramide synthase catalytic subunit AUR1(Saccharomyces cerevisiae S288c)
Pharmacia
Curated by ChEMBL
Pharmacia
Curated by ChEMBL
Affinity DataKi: 0.230nMAssay Description:Inhibition of Saccharomyces cerevisiae SJ21R inositol phosphorylceramide synthase preincubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibition of Candida albicans ATCC 38247 inositol phosphorylceramide synthase preincubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of (S)-N-(2-(1H-pyrrol-1-yl)phenyl)-1-(2-((3H)-1-methyl-1H-benzo[d]imidazol-2-ylthio)acetyl)pyrrolidine-2-carboxamide from human OX2 rec...More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Inhibition of Candida albicans inositol phosphorylceramide synthaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to D4 receptor (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [125I]-OVTA from prairie vole Oxytocin receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Binding affinity to human OT receptorMore data for this Ligand-Target Pair
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataKi: 5.30nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
University Of Strathclyde
Curated by ChEMBL
University Of Strathclyde
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [3H]5CT from 5HT7 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity to human OT receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to rat OX2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity to human OX2 receptorMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to human OTR by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of Candida albicans ATCC 38247 inositol phosphorylceramide synthase preincubated for 30 minsMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity to human OTR by competitive binding assayMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor after 1.5 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]-LVA from prairie vole vasopressin V1A receptor after 72 hrsMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]Oxytocin from human OXTR expressed in CHO cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Texas A&M University
Curated by ChEMBL
Texas A&M University
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Inhibition of wild-type N-terminal TEV cleavage site-fused/His-tagged Mycobacterium tuberculosis H37Rv adenosine kinase expressed in Escherichia coli...More data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Yerkes National Primate Research Center
Curated by ChEMBL
Yerkes National Primate Research Center
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]Oxytocin from human OXTR expressed in CHO cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to human D4 receptor assessed as inhibition constantMore data for this Ligand-Target Pair