Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.28E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataKi: 1.11E+5nMAssay Description:Displacement of [3H]kainate from human GLUK7 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]kainate from rat GLUK6 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUK5 by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA4More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA3More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA2More data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUA1More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUK6More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of glutamate-induced calcium influx in HEK293 cells expressing human GLUK5 by FLIPR assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 3(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataIC50: 2.64E+5nMAssay Description:Displacement of [3H]kainate from human GLUK7 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKd: 402nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.05E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.66E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.88E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.80E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 6.02E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 5.37E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
University Walk
Curated by ChEMBL
University Walk
Curated by ChEMBL
Affinity DataEC50: 2.20E+4nMAssay Description:Induction of calcium influx in HEK293 cells expressing human GLUK5 by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKd: 7.31E+4nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 4.68E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 9.25E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
Affinity DataKd: 1.78E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair