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Report error Found 163 of affinity data for UniProtKB/TrEMBL: P11142
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50442760(CHEMBL2443044)
Affinity DataIC50: 10nMAssay Description:Displacement of N6-(6-amino)hexyl-ATP ATTO-590-ATP from HSC70 (unknown origin) after 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50442759(CHEMBL2443138)
Affinity DataIC50: 10nMAssay Description:Displacement of N6-(6-amino)hexyl-ATP ATTO-590-ATP from HSC70 (unknown origin) after 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50442758(CHEMBL2443139)
Affinity DataIC50: 10nMAssay Description:Displacement of N6-(6-amino)hexyl-ATP ATTO-590-ATP from HSC70 (unknown origin) after 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50442757(CHEMBL2443026)
Affinity DataIC50: 10nMAssay Description:Displacement of N6-(6-amino)hexyl-ATP ATTO-590-ATP from HSC70 (unknown origin) after 18 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataKd:  56nMAssay Description:Binding affinity against HSPA8 (unknown origin) assessed as apparent dissociation constant incubated for 1 hr by colloidal coomassie staining based L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  111nMAssay Description:Binding affinity to human HSPA8 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 130nMAssay Description:Inhibition of HSPA8 (unknown origin) incubated for 1 hr by colloidal coomassie staining based LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM31995(ADP | CHEMBL14830 | Adenosine Diphosphate (ADP))
Affinity DataKd:  260nMAssay Description:Binding affinity to human Hsc70 by isothermal calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085537(CHEMBL3427682)
Affinity DataKd:  280nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50013703(cid_16654696 | diPhosphoric acid [5-(6-amino-purin...)
Affinity DataIC50: 280nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2011
Entry Details
PCBioAssayPDB3D3D Structure (crystal)
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085537(CHEMBL3427682)
Affinity DataKd:  282nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085540(CHEMBL3427679)
Affinity DataKd:  295nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50085540(CHEMBL3427679)
Affinity DataKd:  300nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataKd:  320nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataKd:  324nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443568(CHEMBL3091929)
Affinity DataKd:  400nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184985(CHEMBL3822603)
Affinity DataKd:  457nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184985(CHEMBL3822603)
Affinity DataKd:  460nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50652104(CHEMBL5639838)
Affinity DataKd:  625nMAssay Description:Binding affinity to human recombinant full length HSPA8 (42 to 401 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  660nMAssay Description:Binding affinity to human HSC70 after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32375(adenosine-derived inhibitor (Grp78), 9 | adenosine...)
Affinity DataKd:  720nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32375(adenosine-derived inhibitor (Grp78), 9 | adenosine...)
Affinity DataKd:  724nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443569(CHEMBL3091928)
Affinity DataKd:  900nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443566(CHEMBL3091931)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32372(adenosine-derived inhibitor, 6)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32372(adenosine-derived inhibitor, 6)
Affinity DataKd:  1.45E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443575(CHEMBL3091944)
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  1.61E+3nMAssay Description:Binding affinity to human HSPA8 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443571(CHEMBL3091926)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443574(CHEMBL3091726)
Affinity DataKd:  1.90E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443578(CHEMBL3091941)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443576(CHEMBL3091943)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  2.38E+3nMAssay Description:Binding affinity to human HSC70 Y149A mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443579(CHEMBL3091725)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443570(CHEMBL3091927)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM41998(cid_5351983 | (9Z)-9-[3,3-bis(oxidanyl)prop-2-enyl...)
Affinity DataIC50: 2.73E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2011
Entry Details
PCBioAssay
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184982(CHEMBL3822829)
Affinity DataKd:  2.75E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184982(CHEMBL3822829)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50049820(cid_5153 | 4-Amino-7-(3,4-dihydroxy-5-hydroxymethy...)
Affinity DataKd:  3.24E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50049820(cid_5153 | 4-Amino-7-(3,4-dihydroxy-5-hydroxymethy...)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184984(CHEMBL3823700)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50184984(CHEMBL3823700)
Affinity DataKd:  3.39E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32373(adenosine-derived inhibitor (Grp78), 8 | adenosine...)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32373(adenosine-derived inhibitor (Grp78), 8 | adenosine...)
Affinity DataKd:  3.55E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM41999(MLS-0111617.0001 | 3-(3,4,5-trihydroxy-6-oxo-9-xan...)
Affinity DataIC50: 3.98E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2011
Entry Details
PCBioAssay
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443572(CHEMBL3091728)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443567(CHEMBL3091930)
Affinity DataKd:  5.40E+3nMAssay Description:Binding affinity to human HSC70 after 3 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50281174(CHEMBL4168736)
Affinity DataKd:  5.54E+3nMAssay Description:Binding affinity to human HSC70 Y149W mutant after 2 hrs by fluorescence shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2020
Entry Details Article
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM42000(cid_274125 | 7-methyl-2-[3,4,5-tris(oxidanyl)-6-ox...)
Affinity DataIC50: 5.58E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2011
Entry Details
PCBioAssay
TargetHeat shock cognate 71 kDa protein(Human)
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM32370(adenosine-derived inhibitor (Grp78), 2 | adenosine...)
Affinity DataKd:  6.92E+3nMAssay Description:Binding affinity to human truncated HSC70 NBD (1 to 381 residues) by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2017
Entry Details Article
PubMed
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