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BDBM22862 2-(2-methyl-1H-imidazol-4-yl)ethan-1-amine::2-Methylhistamine

SMILES: Cc1ncc(CCN)[nH]1

InChI Key: InChIKey=XDKYTXBAVJELDQ-UHFFFAOYSA-N

Data: 2 KI 2 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 22862
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H1 receptor (Human)	BDBM22862 (2-(2-methyl-1H-imidazol-4-yl)ethan-1-amine \| 2-Met...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	794	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM22862 (2-(2-methyl-1H-imidazol-4-yl)ethan-1-amine \| 2-Met...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	3.98E+3	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM22862 (2-(2-methyl-1H-imidazol-4-yl)ethan-1-amine \| 2-Met...) Show SMILES Show InChI	GoogleScholar	UniChem		794	-8.65	n/a	n/a	n/a	n/a	n/a	7.4	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM22862 (2-(2-methyl-1H-imidazol-4-yl)ethan-1-amine \| 2-Met...) Show SMILES Show InChI	GoogleScholar	UniChem		794	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair