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BDBM50304527 CHEMBL492677::N4-Benzyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4-diamine

SMILES: CN1CCN(CC1)c1cc(NCc2ccccc2)nc(N)n1

InChI Key: InChIKey=GXRZHULPUGZJMQ-UHFFFAOYSA-N

Data: 2 KI 2 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50304527
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Histamine H4 receptor (Human)	BDBM50304527 (N4-Benzyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	13	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50304527 (N4-Benzyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	63	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50304527 (N4-Benzyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4...) Show SMILES Show InChI	GoogleScholar	UniChem		20	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Histamine H4 receptor (Human)	BDBM50304527 (N4-Benzyl-6-(4-methylpiperazin-1-yl)pyrimidine-2,4...) Show SMILES Show InChI	GoogleScholar	UniChem		98	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair