BDBM50328476 1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetrazol-5-yl)methyl)-1H-indol-3-yl)piperidin-1-yl)ethyl)imidazolidin-2-one::CHEMBL1259188

SMILES Cn1nnc(Cc2ccc3n(cc(C4CCN(CCN5CCNC5=O)CC4)c3c2)-c2ccc(F)cc2)n1

InChI Key InChIKey=FGHKCRNDQSRICR-UHFFFAOYSA-N

Data  4 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50328476   

TargetAlpha-1B adrenergic receptor(C.H.O.)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]prozosin from hamster cloned alpha1b receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prozosin from bovine cloned alpha1a receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]prozosin from rat cloned alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50328476(1-(2-(4-(1-(4-fluorophenyl)-5-((2-methyl-2H-tetraz...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]prozosin from human cloned dopamine D2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed