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BDBM66983 6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazepine;hydrochloride::6-chloro-3-methyl-1,2,4,5-tetrahydro-3-benzazepine;hydrochloride::CHEMBL123349::MLS002172470::SKF 86466::SKF-86466 hydrochloride::SMR001254100::cid_10220250

SMILES: CN1CCc2cccc(Cl)c2CC1

InChI Key: InChIKey=RSRUDTPYRBLHEO-UHFFFAOYSA-N

Data: 16 KI  1 EC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 17 hits for monomerid = 66983   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Bcl-2-like protein 11


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
n/an/an/an/a>3.50E+5n/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2B adrenergic receptor


(Rat)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
1.80n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2A adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
2.40n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2C adrenergic receptor


(OK)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
2.70n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor


(Rat)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
7.90n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2A adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
9.40n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2A adrenergic receptor


(Guinea pig)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
13n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2B adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
16n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
17n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2C adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
20n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-2B adrenergic receptor


(Dog)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
42n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
5-hydroxytryptamine receptor 1A


(Rat)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
100n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-1D adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
126n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-1A adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
449n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-1B adrenergic receptor


(Human)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
485n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-1A adrenergic receptor


(Rabbit)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
900n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Alpha-1A adrenergic receptor


(Dog)
BDBM66983
PNG
(MLS002172470 | SMR001254100 | SKF-86466 hydrochlor...)
GoogleScholar
UniChem
1.10E+3n/an/an/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair