TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute
Curated by PDSP Ki Database
Barrow Neurological Institute
Curated by PDSP Ki Database
Affinity DataKi: 0.0700nMAssay Description:Inhibitory activity against human tryptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute
Curated by PDSP Ki Database
Barrow Neurological Institute
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory activity against human tryptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.850nMAssay Description:Inhibition of trypsin in human mast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Inhibition of trypsin in human mast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to Cav3.3 alpha1iMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute
Curated by PDSP Ki Database
Barrow Neurological Institute
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute
Curated by PDSP Ki Database
Barrow Neurological Institute
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Antagonist activity at Cav3.3 alpha1i expressed in HEK293 cells at -100 mV by standard voltage-clamp electrophysiology assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition plasmin in human mast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Barrow Neurological Institute
Curated by PDSP Ki Database
Barrow Neurological Institute
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair