TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in the presence of pig liver esterase, in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Compound was evaluated in vitro for the ability to inhibit HIV-protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 100 mg/kgMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory constant of the compound was tested angiotensin converting enzymeMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in the presence of pig liver esterase, in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Compound was evaluated in vitro for the ability to inhibit HIV-protease.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in the presence of pig liver esterase, in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in the presence of pig liver esterase, in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in the presence of pig liver esterase, in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 50 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 50 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 50 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 50 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 25 mg/kgMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Evaluated for its activity to inhibit rat liver 2,3-oxidosqualene-lanosterol cyclase, activity expressed as KiMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 50 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:In vitro inhibitory activity against human neutrophil elastase was determined at a dose of 45 mg/kgMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 195nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 261nMAssay Description:In vitro inhibitory activity against human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Evaluated for its activity to inhibit rat liver 2,3-oxidosqualene-lanosterol cyclase, activity expressed as KiMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:In vitro inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Binding affinity of the compound against Angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: 1.50E+5nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+5nMAssay Description:Binding affinity of the compound against neutral endopeptidaseMore data for this Ligand-Target Pair
TargetNeutrophil elastase(Homo sapiens (Human))
Marion Merrell Dow Research Institute
Curated by ChEMBL
Marion Merrell Dow Research Institute
Curated by ChEMBL
Affinity DataKi: >5.00E+5nMAssay Description:Binding affinity of the compound for purified Human neutrophil elastase was determined in vitro.More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Concentration required to inhibit rat liver 2,3-oxidosqualene-lanosterol cyclase (OSC)More data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Concentration required to inhibit rat liver 2,3-oxidosqualene-lanosterol cyclaseMore data for this Ligand-Target Pair