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Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
361 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-2
  • ALK tyrosine kinase receptor
  • Actin-related protein 2
  • Activin receptor type-1
  • Activin receptor type-1B
  • Aurora kinase A/B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • BR serine/threonine-protein kinase 1
  • BR serine/threonine-protein kinase 2
  • BRAF/CRAF
  • Beta-adrenergic receptor kinase 2
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Bone morphogenetic protein receptor type-2
  • CAMK2A
  • CAMK2B
  • CDC7/Cyclin B1
  • CDK2/CycE
  • CDK2/Cyclin A1
  • CDK3/E
  • CDK4/Cyclin D3
  • CDK6/CycD3
  • CDK7/Cyclin H/MNAT1
  • CDKL2
  • CaM kinase I alpha
  • CaM kinase I delta
  • CaM kinase I gamma
  • CaM kinase II
  • CaM kinase IV
  • CaM-kinase kinase alpha
  • CaM-kinase kinase beta
  • Calcium/calmodulin-dependent protein kinase type 1B
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Casein kinase I
  • Casein kinase I isoform delta
  • Casein kinase I isoform gamma-3
  • Casein kinase II subunit alpha
  • Casein kinase II subunit alpha 3
  • Cereblon/BCR/ABL
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-Y
  • Cyclin-dependent kinase 12
  • Cyclin-dependent kinase 13/Cyclin-K
  • Cyclin-dependent kinase 18
  • Cyclin-dependent kinase-like 1
  • Cyclin-dependent kinase-like 3
  • Cyclin-dependent kinase-like 4
  • Cytoplasmic tyrosine-protein kinase BMX
  • DNA-PK/Ku70/Ku85
  • Death-associated protein kinase 1
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Discoidin domain-containing receptor 2
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
  • Dual specificity mitogen-activated protein kinase kinase; MEK1/2
  • Dual specificity protein kinase CLK1/CLK4
  • Dual specificity protein kinase CLK2
  • Dual specificity protein kinase CLK3
  • Dual specificity protein kinase TTK
  • Dual specificity tyrosine-phosphorylation-regulated kinase 1B
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Dual-specificity tyrosine-phosphorylation regulated kinase 2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 3
  • EPHB1
  • Ephrin receptor
  • Ephrin type-A receptor 2
  • Ephrin type-A receptor 3 (EPHA3)
  • Ephrin type-A receptor 7
  • Ephrin type-B receptor 3 (EPHB3)
  • Ephrin type-B receptor 4
  • Epidermal growth factor receptor
  • Eukaryotic elongation factor 2 kinase
  • Eukaryotic translation initiation factor 2-alpha kinase 1
  • Eukaryotic translation initiation factor 2-alpha kinase 4
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
  • G protein-coupled receptor kinase 5
  • G protein-coupled receptor kinase 6
  • G protein-coupled receptor kinase 7
  • G-protein coupled receptor kinase 2
  • Glucokinase/Glucokinase regulatory protein
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 1
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Homeodomain-interacting protein kinase 3
  • Homeodomain-interacting protein kinase 4
  • Inhibitor of NF-kappa-B kinase alpha/beta
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Insulin receptor-related protein
  • Insulin-like growth factor I receptor
  • Interferon-induced, double-stranded RNA-activated protein kinase
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • LIM domain kinase 2
  • Leucine-rich repeat serine/threonine-protein kinase 2
  • Leukocyte tyrosine kinase receptor
  • MAP kinase-activated protein kinase 3
  • MAP kinase-interacting serine/threonine-protein kinase 1/2
  • MAP/microtubule affinity-regulating kinase 2
  • MAP/microtubule affinity-regulating kinase 3
  • MAP/microtubule affinity-regulating kinase 4
  • MAPK/MAK/MRK overlapping kinase
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Macrophage-stimulating protein receptor
  • Mammalian target of Rapamycin (mTORC1)
  • Mast/stem cell growth factor receptor Kit
  • Maternal embryonic leucine zipper kinase
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 10/Receptor-interacting serine/threonine-protein kinase 1
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 14
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase kinase kinase 10
  • Mitogen-activated protein kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase 5
  • Mitogen-activated protein kinase kinase kinase 7
  • Mitogen-activated protein kinase kinase kinase 9
  • Mitogen-activated protein kinase kinase kinase kinase 1
  • Mitogen-activated protein kinase kinase kinase kinase 3
  • Mitogen-activated protein kinase kinase kinase kinase 4
  • Mitogen-activated protein kinase kinase kinase kinase 5
  • Mixed lineage kinase 7
  • Muscle, skeletal receptor tyrosine protein kinase
  • Myosin light chain kinase, smooth muscle
  • Myosin-IIIB
  • Myotonin-protein kinase
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • NUAK family SNF1-like kinase 2
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • PAS domain-containing serine/threonine-protein kinase
  • PKC alpha and beta-2
  • PRP4 kinase (PRP4)
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Pancreatic endoplasmic reticulum kinase (PERK)
  • Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
  • Phosphorylase kinase
  • Platelet-derived growth factor receptor
  • Platelet-derived growth factor receptor beta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase C, PKC; classical/novel
  • Protein kinase N1
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Pyruvate dehydrogenase kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • RAF serine/threonine protein kinase
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Rhodopsin kinase
  • Ribosomal protein S6 kinase
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 4
  • Ribosomal protein S6 kinase alpha 6
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine-protein kinase ATM
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 10
  • Serine/threonine-protein kinase 11
  • Serine/threonine-protein kinase 16
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 17B (STK17B)
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase 24
  • Serine/threonine-protein kinase 25
  • Serine/threonine-protein kinase 32A
  • Serine/threonine-protein kinase 32B
  • Serine/threonine-protein kinase 32C
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 35
  • Serine/threonine-protein kinase 38-like
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Aurora-C
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase DCLK2
  • Serine/threonine-protein kinase DCLK3
  • Serine/threonine-protein kinase ICK
  • Serine/threonine-protein kinase MAK
  • Serine/threonine-protein kinase MRCK beta
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase NEK2
  • Serine/threonine-protein kinase NEK6
  • Serine/threonine-protein kinase NEK7
  • Serine/threonine-protein kinase NEK9
  • Serine/threonine-protein kinase NIM1
  • Serine/threonine-protein kinase Nek1
  • Serine/threonine-protein kinase Nek11
  • Serine/threonine-protein kinase Nek3
  • Serine/threonine-protein kinase Nek4
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PAK7
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PRKX
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase SBK1
  • Serine/threonine-protein kinase SIK1
  • Serine/threonine-protein kinase SIK2
  • Serine/threonine-protein kinase SIK3
  • Serine/threonine-protein kinase SRPK1
  • Serine/threonine-protein kinase SRPK2
  • Serine/threonine-protein kinase SRPK3
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase Sgk2
  • Serine/threonine-protein kinase Sgk3
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TAO2
  • Serine/threonine-protein kinase TAO3
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase ULK1
  • Serine/threonine-protein kinase ULK2
  • Serine/threonine-protein kinase ULK3
  • Serine/threonine-protein kinase VRK1
  • Serine/threonine-protein kinase VRK2
  • Serine/threonine-protein kinase WEE1
  • Serine/threonine-protein kinase WNK1
  • Serine/threonine-protein kinase WNK2
  • Serine/threonine-protein kinase WNK3
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Serine/threonine-protein kinase pim-3
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase tousled-like 1
  • Serine/threonine-protein kinase tousled-like 2
  • Serine/threonine-protein kinase/endoribonuclease IRE1 Alpha
  • TGF-beta receptor type II
  • TGF-beta receptor type-1
  • TRAF2- and NCK-interacting kinase
  • Tau-tubulin kinase 1
  • Tau-tubulin kinase 2
  • Testis-specific serine/threonine-protein kinase 1
  • Testis-specific serine/threonine-protein kinase 2
  • Testis-specific serine/threonine-protein kinase 3
  • Testis-specific serine/threonine-protein kinase 4
  • Transcription initiation factor TFIID subunit 1-like
  • Transient receptor potential cation channel subfamily M member 7
  • Tribbles homolog 2
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase FER
  • Tyrosine-protein kinase FES
  • Tyrosine-protein kinase FRK
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase TXK
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • Wee1-like protein kinase 2
  • cAMP-dependent protein kinase (PKA)
  • cGMP-dependent protein kinase 1 beta
  • cGMP-dependent protein kinase 2
  • mTOR/FKBP12A/FKBP12B
  • myosin light chain kinase 2
  • p110α/p85α
  • p110β/p85α
  • p21-Activated kinase 3 (PAK3)
  • p38 MAP kinase alpha/beta
  • p38 delta/gamma
  • CHEMBL4438748