Protein Targets in BindingDB are mapped to TrEMBL entries based on 100% sequence identity, with the program BLAST. Note that the BindingDB and TrEMBL sequences do not need to be exactly the same length to meet this criterion. TrEMBL's Secondary Accession IDs are obsolete IDs for the same protein, and are included here because older papers may use these IDs.
- Primary IDUniProt Recommended NameBindingDB NameAffinity Link(s)ArticlesDownloads
- DNA ligasePolydeoxyribonucleotide synthase [ATP]IC50=11
- Clamp loader small subunitClamp loader small subunitITC=4
- DNA-directed DNA polymeraseDNA polymeraseIC50=9
- Serpin peptidase inhibitor, clade E (Nexin, plasminogen activator inhibitor type 1), member 1, isoform CRA_bPAI
- Serine/threonine-protein kinasePim-2h
- Emopamil binding proteinCholestenol Delta-isomerase
- Phosphoribosyl pyrophosphate synthetase-associated protein 2, isoform CRA_aPhosphoribosyl pyrophosphate synthetase-associated protein 2Ki=3
- B-cell CLL/lymphoma 9, isoform CRA_aBCL9
- Mitogen-activated protein kinaseNLK
- Heme carrier protein 1, isoform CRA_aG21
- Mitogen-activated protein kinaseMitogen-activated protein kinase 7
- Histone deacetylase 6, isoform CRA_cHistone deacetylase 6 (HDAC6)
- GalectinGalectin-9Kd=72
- TAO kinase 1, isoform CRA_aSerine/threonine-protein kinase TAO1
- EPH receptor A2, isoform CRA_aECK
- AKT1 substrate 1 (Proline-rich), isoform CRA_a40 kDa proline-rich AKT substrateIC50=68
- Phospholipase A2, group IVC (Cytosolic, calcium-independent), isoform CRA_dPhospholipase A2 group IVCIC50=5
- Sphingosine kinase 2, isoform CRA_cSPK 2
- FCGRTIgG receptor FcRn large subunit p51
- Plasminogen activator, urokinase, isoform CRA_aUrokinase
- Chromosome 10 open reading frame 70, isoform CRA_bCDGSH iron-sulfur domain-containing protein 1
- Sirtuin (Silent mating type information regulation 2 homolog) 1 (S. cerevisiae), isoform CRA_aSIRT1
- Peptidyl-prolyl cis-trans isomeraseCyclophilin FKd=112
- Epididymis secretory sperm binding proteinVDAC-2Kd=1
- Receptor (TNFRSF)-interacting serine-threonine kinase 1, isoform CRA_aReceptor-interacting protein 1
- Eukaryotic translation initiation factor 2-alpha kinase 1, isoform CRA_aEukaryotic translation initiation factor 2-alpha kinase 1
- Serine/threonine-protein kinase PLKPolo-Like Kinase 2
- Elongation of very long chain fatty acids protein 2Elongation of very long chain fatty acids protein 2IC50=4
- Thiopurine S-methyltransferase, isoform CRA_dThiopurine S-methyltransferase
- PRP4 pre-mRNA processing factor 4 homolog B (Yeast), isoform CRA_aPRP4 kinase
- NAD-dependent protein deacylase sirtuin-5, mitochondrialNAD-dependent protein deacetylase sirtuin-5 (SIRT5)
- HCG37731, isoform CRA_cRAD1
- Amino acid transporterExcitatory Amino Acid EAAT1
- NAD kinase, isoform CRA_aNAD kinase
- AdenosylhomocysteinaseAHCYL1IC50=5
- Epididymis secretory sperm binding proteinRho-related GTP-binding protein RhoCIC50=34
- Hydroxy-delta-5-steroid dehydrogenase, 3 beta-and steroid delta-isomerase 2, isoform CRA_a3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type IIIC50=4
- Solute carrier family 16 (Monocarboxylic acid transporters), member 1, isoform CRA_bMonocarboxylate transporter 1
- Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1B, isoform CRA_aDYRK1B
- Non-specific serine/threonine protein kinaseSerine/threonine-protein kinase PAK 4
- Glycogen synthase kinase 3 alpha, isoform CRA_aGlycogen synthase kinase-3 alpha (GSK3A)
- Transforming growth factor betaTransforming growth factor beta-1IC50=7
- Serine/threonine-protein phosphatasePP5
- Rho guanine nucleotide exchange factor (GEF) 1, isoform CRA_e115 kDa guanine nucleotide exchange factorIC50=1
- Egl nine homolog 2 (C. elegans), isoform CRA_bProlyl hydroxylase domain-containing protein 1 (PHD1)IC50=629
- SUMO-1 activating enzyme subunit 1, isoform CRA_bSUMO1 activating enzyme subunit 1IC50=257
- ATP-dependent 6-phosphofructokinasePhosphofructokinase muscle typeEC50=1
- Protein kinase, AMP-activated, gamma 1 non-catalytic subunit, isoform CRA_aAMPK alpha2/beta2/gamma1
- Nuclear receptor subfamily 4, group A, member 1, isoform CRA_dnuclear receptor subfamily 4, group A, member 1
- Cathepsin L2, isoform CRA_aCathepsin (V and K)
- UDP-glucose ceramide glucosyltransferase, isoform CRA_aGCSIC50=262
- V-raf murine sarcoma 3611 viral oncogene homolog, isoform CRA_bProto-oncogene A-Raf-1IC50=22
- Testicular secretory protein Li 63Ubiquitin-like modifier-activating enzyme 1IC50=130
- ELK1, member of ETS oncogene family, isoform CRA_aETS domain-containing protein (Elk1)IC50=5
- G protein-coupled receptor kinaseBeta-adrenergic receptor kinase 2IC50=8
- X-box binding protein 1, isoform CRA_bXBP1
- Protein-tyrosine sulfotransferaseProtein-tyrosine sulfotransferase 2IC50=5
- LIM domain kinase 2, isoform CRA_aLIM domain kinase 2
- Tyrosine 3-monooxygenase/tryptophan 5-monooxygenase activation protein, eta polypeptide, isoform CRA_bYWHA1Kd=1
- Potassium inwardly-rectifying channel, subfamily J, member 4, isoform CRA_aHIRK2IC50=6
- Myosin, heavy polypeptide 9, non-muscle, isoform CRA_aCellular myosin heavy chain, type AIC50=1
- Sterol regulatory element binding transcription factor 2, isoform CRA_aSterol regulatory element-binding protein 2IC50=30
- Chromobox homolog 7, isoform CRA_bChromobox protein homolog 7 (CBX7)
- ATP-citrate synthaseATP-citrate synthase
- Insulin-like growth factor binding protein 4, isoform CRA_aInsulin-like growth factor binding protein 4Ki=2
- Guanine deaminaseGAH
- Tyrosine-protein kinaseSpleen Tyrosine Kinase
- Cathepsin L, isoform CRA_aMEP
- Serine palmitoyltransferase, long chain base subunit 1, isoform CRA_aSerine-palmitoyl-CoA transferase 1IC50=1
- B-cell CLL/lymphoma 2, isoform CRA_aApoptosis regulator Bcl-2/Bcl-2 homologous antagonist/killer
- Lipase, endothelial, isoform CRA_aELIC50=1406
- Transcription factor 4, isoform CRA_bSEF-2
- von Hippel-Lindau tumor suppressor isoform 2 (Fragment)pVHL
- Thyroid hormone nuclear receptor beta variant 1c-erbA-2
- Ubiquitin-conjugating enzyme E2E 1 (UBC4/5 homolog, yeast), isoform CRA_aE2 ubiquitin-conjugating enzyme E1IC50=125
- TransporterSolute carrier family 6 member 1
- Testicular tissue protein Li 224WDR48
- Catenin (Cadherin-associated protein), beta 1, 88kDa, isoform CRA_aCatenin beta-1
- Protein kinase cAMP-dependent regulatory type II alpha isoform 2 (Fragment)PKR2Kd=11
- Mitogen-activated protein kinase-activated protein kinase 3, isoform CRA_aMAPKAPK-3
- Hyaluronidase (Fragment)Hyaluronoglucosaminidase-1IC50=22
- SNF related kinase, isoform CRA_aSNF-related serine/threonine-protein kinaseKd=72
- Ubiquitin carboxyl-terminal hydrolaseUbiquitin carboxyl-terminal hydrolase BAP1 (BRCA1-associated protein 1) (Cerebral protein 6).IC50=42
- Poly [ADP-ribose] polymerasePARP3IC50=39
- Abhydrolase domain containing 6, isoform CRA_aABHD6
- Epididymis secretory sperm binding proteinh12
- Protein kinase C delta typeProtein kinase C, PKC; classical/novel
- Scm-like with four mbt domains 1, isoform CRA_bhSFMBTIC50=56
- DeoxyribonucleaseLSDIC50=5
- Bis(5'-adenosyl)-triphosphataseDinucleosidetriphosphataseKi=29
- Cathepsin B, isoform CRA_aCathepsin B heavy chain
- Double-strand break repair proteinMRE11AIC50=2
- PannexinPANX1IC50=1
- Dopamine receptor D2, isoform CRA_cDopamine D2A
- Zinc finger and BTB domain containing 16 isoform 1Zinc finger and BTB domain-containing protein 16IC50=17
- Serine-protein kinase ATMAtaxia telangiectasia mutated
- Beta-site APP-cleaving enzyme 1, isoform CRA_dAspartyl protease 2
- SNF1-like kinase 2, isoform CRA_cSerine/threonine-protein kinase SIK2
- Solute carrier family 37 (Glycerol-6-phosphate transporter), member 4, isoform CRA_aTRG-19IC50=13
- Dopamine receptor D2, isoform CRA_bDopamine D2 S receptor
- Friend leukemia virus integration 1, isoform CRA_aProto-oncogene Fli-1
- Degenerative spermatocyte homolog 1, lipid desaturase (Drosophila), isoform CRA_aSphingolipid delta(4)-desaturase DES1IC50=2
- Acyl-Coenzyme A binding domain containing 3, isoform CRA_aGolgi resident protein GCP60Ki=4
- ADP-ribosylation factor 1, isoform CRA_aADP-ribosylation factor 1Kd=1
- Geranylgeranyl diphosphate synthase 1, isoform CRA_aGeranylgeranyl pyrophosphate synthetase
- Poly [ADP-ribose] polymeraseADPRT
- Muscarinic acetylcholine receptorRecName: Full=Muscarinic acetylcholine receptor M3
- Epididymis secretory sperm binding protein (Fragment)HSP60/HSP10IC50=214
- Isocitrate dehydrogenase [NADP]Oxalosuccinate decarboxylase
- Small ubiquitin-related modifierSmall ubiquitin-related modifier 1IC50=2
- Alkaline phosphataseAlkaline phosphatase, intestinal
- Serine/threonine kinase 25 (STE20 homolog, yeast), isoform CRA_a (Fragment)YSK1
- Catenin, beta interacting protein 1, isoform CRA_aICATIC50=10
- Enolase 1, (Alpha), isoform CRA_aC-myc promoter-binding proteinIC50=3
- DNA polymeraseDNA polymerase delta subunit 1IC50=17
- Protein-S-isoprenylcysteine O-methyltransferaseIsoprenylcysteine carboxyl methyltransferase
- Kallikrein 7 (Chymotryptic, stratum corneum), isoform CRA_bKallikrein 7
- Kallikrein 2, prostatic, isoform CRA_aKallikrein 2
- Kallikrein 6 (Neurosin, zyme), isoform CRA_bKallikrein 6
- Malate dehydrogenaseMalate dehydrogenase, mitochondrial
- Kallikrein 12, isoform CRA_cKallikrein-12Ki=3
- Kallikrein 14, isoform CRA_aKallikrein-14
- Formyl peptide receptor-like 1, isoform CRA_aLXA4 receptor
- Epsin 1, isoform CRA_aEH domain-binding mitotic phosphoproteinIC50=2
- Epididymis secretory sperm binding protein2.3.2.-Kd=1
- Ceramide kinase, isoform CRA_bhCERK
- Bromodomain containing 1, isoform CRA_bBR140-like protein
- HCG2044796, isoform CRA_aCPTI-MIC50=21
- HCG16873, isoform CRA_aCKB
- Solute carrier family 43, member 1, isoform CRA_bL-type amino acid transporter 3IC50=3
- BCL2-antagonist of cell death, isoform CRA_cBcl-XL/Bcl-2-associated death promoter
- Non-specific serine/threonine protein kinaseGCK
- Histone acetyltransferaseHistone acetyltransferase KAT5IC50=17
- HCG1810791, isoform CRA_bPotassium channel subfamily K member 4EC50=1
- Mitogen-activated protein kinase kinase kinaseMLK3
- Carnitine palmitoyltransferase 1A (Liver), isoform CRA_aCPTI-L
- 7-dehydrocholesterol reductase isoform 1Sterol Delta(7)-reductase
- Folate receptor 1 (Adult), isoform CRA_aFolate receptor 1
- Pyrimidinergic receptor P2Y, G-protein coupled, 6, isoform CRA_bP2Y6
- Serpin peptidase inhibitor, clade H (Heat shock protein 47), member 1, (Collagen binding protein 1), isoform CRA_aCollagen-binding protein 1IC50=4
- Prolylcarboxypeptidase (Angiotensinase C), isoform CRA_aProlylcarboxypeptidase (PRCP)
- Non-specific serine/threonine protein kinasePAK-1
- Adenylosuccinate synthetase isozyme 2Adenylosuccinate synthetase isozyme 2IC50=3
- Ubiquitin specific peptidase 8, isoform CRA_aUbiquitin carboxyl-terminal hydrolase 8IC50=7
- Cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aP-450AROM
- ADAM metallopeptidase domain 10, isoform CRA_bDisintegrin and metalloproteinase domain-containing protein 10 (ADAM10)
- HCG2004507, isoform CRA_aCasein kinase I isoform gamma-1
- Mitogen-activated protein kinase kinase 5, isoform CRA_aMAPKK 5
- Mothers against decapentaplegic homologmothers against decapentaplegic homolog 3IC50=66
- Poly [ADP-ribose] polymerasePARP6IC50=6
- Dipeptidyl-peptidase 8, isoform CRA_fDPP8
- Death-associated protein kinase 2, isoform CRA_bDeath-associated protein kinase 2
- CDK-activating kinase assembly factor MAT1CDK-activating kinase assembly factor MAT1 (CDK7/H/MAT1)IC50=1
- GalectinGalectin-3
- ArginaseArginase II
- PresenilinGamma-Secretase Subunit Presenilin-1
- Protein phosphatase 1A (Formerly 2C), magnesium-dependent, alpha isoform, isoform CRA_aProtein phosphatase 1AIC50=16
- Serine palmitoyltransferase, long chain base subunit 2, isoform CRA_aSerine-palmitoyl-CoA transferase 2IC50=14
- Inositol 1,3,4-triphosphate 5/6 kinase, isoform CRA_aInositol TriphosphateKi=2
- Cyclin K, isoform CRA_cCyclin-KIC50=36
- Tyrosyl-DNA phosphodiesterase 1, isoform CRA_aTyrosyl-DNA phosphodiesterase 1
- CDC42 binding protein kinase beta (DMPK-like), isoform CRA_aMyotonic dystrophy kinase-related CDC42-binding kinase beta
- Matrix metallopeptidase 2 (Gelatinase A, 72kDa gelatinase, 72kDa type IV collagenase), isoform CRA_aMatrix metalloproteinase-2
- TransporterNoradrenaline Transporter (NET)
- Matrix metallopeptidase 15 (Membrane-inserted), isoform CRA_aMembrane-type matrix metalloproteinase 2
- Core-binding factor, beta subunit, isoform CRA_bCore-binding factor subunit beta (CBFB)IC50=36
- Peptide deformylasePolypeptide deformylase
- HCG2026222, isoform CRA_cChymotrypsin-like protease CTRL-1IC50=22
- Dihydrouridine synthase 2-like, SMM1 homolog (S. cerevisiae), isoform CRA_aUp-regulated in lung cancer protein 8IC50=1
- SFRS protein kinase 2, isoform CRA_bSRSF protein kinase 2 N-terminal
- Protein kinase, cAMP-dependent, regulatory, type II, beta, isoform CRA_acAMP-dependent protein kinase type II-beta regulatory subunit
- Nicotinamide phosphoribosyltransferaseNicotinamide phosphoribosyltransferase
- Phosphoinositide-3-kinase, catalytic, gamma polypeptide, isoform CRA_aPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/gamma isoform
- Protein arginine N-methyltransferase[Myelin basic protein]-arginine N-methyltransferase PRMT7
- Met proto-oncogene (Hepatocyte growth factor receptor), isoform CRA_aHepatocyte growth factor receptor (HGFR)IC50=13
- Cystic fibrosis transmembrane conductance regulatorChannel conductance-controlling ATPase
- POT1 protection of telomeres 1 homolog (S. pombe), isoform CRA_bProtection of telomeres protein 1IC50=4
- Met proto-oncogene (Hepatocyte growth factor receptor), isoform CRA_cc-Met kinase
- Aldo-keto reductase family 1, member B1 (Aldose reductase), isoform CRA_aAR
- Endothelial differentiation, sphingolipid G-protein-coupled receptor, 5, isoform CRA_aSphingosine 1-phosphate receptor
- CDC37 cell division cycle 37 homolog (S. cerevisiae), isoform CRA_aHsp90 co-chaperone
- Kelch-like ECH-associated protein 1, isoform CRA_aKelch-like ECH-associated protein 1
- Low density lipoprotein receptor (Familial hypercholesterolemia), isoform CRA_bLow-density lipoprotein receptorEC50=17
- Tyrosine-protein kinaseNon-receptor tyrosine-protein kinase TYK2 (TYK2)
- Deoxyribonuclease II, lysosomal, isoform CRA_aDNase II alphaKi=1
- Protein kinase, cAMP-dependent, catalytic, alpha, isoform CRA_ccAMP-dependent protein kinase catalytic subunit alpha
- Tyrosine-protein kinaseJanus kinase 3 (JAK3)
- Endothelial differentiation, lysophosphatidic acid G-protein-coupled receptor, 4, isoform CRA_aLysophosphatidic acid receptor 2
- Testis secretory sperm-binding protein Li 205aTSSK-6IC50=1
- Solute carrier family 34 (Sodium phosphate), member 1, isoform CRA_bSLC34A1
- Proto-oncogene tyrosine-protein kinase receptor RetRET51
- COP9 constitutive photomorphogenic homolog subunit 5 (Arabidopsis), isoform CRA_aCOP9 signalosome complex subunit 5 (Csn5)IC50=66
- Transcription elongation factor B (SIII), polypeptide 1 (15kDa, elongin C), isoform CRA_aEloC
- Uncharacterized proteinProteasome assembly chaperone 3IC50=1
- Non-specific serine/threonine protein kinaseCytokine-independent survival kinase
- G protein-coupled receptor 30, isoform CRA_aG-protein-coupled receptor (GPR30 )
- Solute carrier family 2, (Facilitated glucose transporter) member 8, isoform CRA_aGlucose transporter type 8IC50=5
- Cyclin-dependent kinase 9 (CDC2-related kinase), isoform CRA_aTat-associated kinase complex catalytic subunit
- NIMA (Never in mitosis gene a)-related kinase 6, isoform CRA_bSerine/threonine-protein kinase NEK6
- Frequenin homolog (Drosophila), isoform CRA_aFREQKd=2
- Solute carrier family 27 (Fatty acid transporter), member 4, isoform CRA_aFatty acid transport protein 4IC50=48
- Protein kinase N3, isoform CRA_aProtein-kinase C-related kinase 3IC50=1
- Tyrosine-protein kinasetyrosine-protein kinase ABL1 isoform a
- Prostaglandin D2 synthase 21kDa (Brain), isoform CRA_aPGD2Ki=5
- Bromodomain containing 3, isoform CRA_aBromodomain-containing protein 3 (BRD3)
- 1-acyl-sn-glycerol-3-phosphate acyltransferase1-acylglycerol-3-phosphate O-acyltransferase betaIC50=131
- Protein tyrosine phosphatase type IVA, member 1, isoform CRA_aProtein tyrosine phosphatase type IVA 1IC50=20
- Protein disulfide-isomeraseCellular thyroid hormone-binding protein
- Solute carrier family 16 (Monocarboxylic acid transporters), member 3, isoform CRA_aMCT4IC50=397
- DEAD (Asp-Glu-Ala-Asp) box polypeptide 48, isoform CRA_aEukaryotic translation initiation factor 4A isoform 3
- POU domain proteinOctamer-binding transcription factor 1IC50=2
- Mitochondrial pyruvate carrierMPC2IC50=2
- Discoidin domain receptor family, member 2, isoform CRA_aDiscoidin domain-containing receptor 2
- Regulator of G-protein signalling 4, isoform CRA_aRegulator of G-protein signaling 4 (RGS4)
- HCG2024989, isoform CRA_a3-keto-steroid reductaseIC50=3
- Solute carrier family 19 (Thiamine transporter), member 2, isoform CRA_a (Fragment)ThTr-1Ki=2
- Serpin peptidase inhibitor, clade C (Antithrombin), member 1, isoform CRA_aAntithrombin-III
- Ubiquitin-conjugating enzyme E2T (Putative), isoform CRA_aUbiquitin carrier protein TKd=1
- Polyadenylate-binding proteinpolyadenylate-binding protein 1IC50=611
- ATPase family, AAA domain containing 2, isoform CRA_cATAD2
- Potassium channel subfamily K memberPotassium channel subfamily K member 9IC50=117
- Muscarinic acetylcholine receptorCHRM5
- NADH dehydrogenase (Ubiquinone) 1 alpha subcomplex, assembly factor 1, isoform CRA_aNADH dehydrogenase [ubiquinone] 1 alpha subcomplex assembly factor 1
- ST3 beta-galactoside alpha-2,3-sialyltransferase 1, isoform CRA_aCMP-N-acetylneuraminate-beta-galactosamide-alpha-2,3-sialyltransferase 1IC50=3
- Myc proto-oncogene proteinMyc proto-oncogene protein
- Non-specific serine/threonine protein kinasePAK6
- Gamma-aminobutyric acid (GABA) A receptor, alpha 2, isoform CRA_aGamma-aminobutyric acid receptor subunit alpha-2 (GABRA2)
- Microtubule-associated proteinMicrotubule-associated protein tau
- FYVE, RhoGEF and PH domain containing 1 (Faciogenital dysplasia), isoform CRA_aRho/Rac guanine nucleotide exchange factorKi=1
- NADH dehydrogenase (Ubiquinone) 1 alpha subcomplex, 4, 9kDa, isoform CRA_bNADH-ubiquinone oxidoreductase MLRQ subunitIC50=4
- Aryl hydrocarbon receptor, isoform CRA_aAhR
- Microtubule-associated proteinMicrotubule-associated protein Tau isoform 2N4R (Tau 2N4R)IC50=64
- Aquaporin 1 (Channel-forming integral protein, 28kDa)Aquaporin-1 (AQP1)IC50=6
- Caspase recruitment domain family, member 4nucleotide-binding oligomerization domain containing 1
- Cell division cycle 2-like 5 (Cholinesterase-related cell division controller), isoform CRA_aCell division protein kinase 13Kd=72
- Phospholipase A(2)Phosphatidylcholine 2-acylhydrolaseIC50=595
- Cell division cycle 42 (GTP binding protein, 25kDa), isoform CRA_aG25K GTP-binding protein
- Alkaline phosphatasetissue-nonspecific alkaline phosphatase precursor
- Mitogen-activated protein kinase kinase kinase 2, isoform CRA_aMitogen-activated protein kinase kinase kinase 2
- Cannabinoid receptor 2 (Macrophage), isoform CRA_aCB2
- Beta-hexosaminidaseHexosaminidase subunit B
- Glutaredoxin (Thioltransferase), isoform CRA_cGlutaredoxin-1 (GRX-1)Ki=1
- 3-hydroxy-3-methylglutaryl coenzyme A reductaseHMG-CoA reductase
- Polymerase (DNA directed) kappa, isoform CRA_bDNA polymerase kappa
- Coagulation factor II (Thrombin) receptor, isoform CRA_aPAR-1
- Betaine-homocysteine methyltransferase 2, isoform CRA_cBetaine--homocysteine S-methyltransferase 2
- Solute carrier organic anion transporter family memberSodium-independent organic anion transporterKi=2
- Solute carrier organic anion transporter family memberThromboxane B2
- Branched-chain-amino-acid aminotransferaseBranched-chain-amino-acid transferaseIC50=31
- ATP-dependent DNA helicaseRecQ protein-like 1IC50=5
- ATP-binding cassette, sub-family C (CFTR/MRP), member 9, isoform CRA_bATP-binding cassette transporter sub-family C member 9EC50=56
- Microsomal glutathione S-transferase 1, isoform CRA_aGlutathione S-transferase (GST)
- Mitogen-activated protein kinase kinase kinase 12DLK
- Heterogeneous nuclear ribonucleoprotein A1, isoform CRA_bhnRNP core protein A1Kd=1
- TetraspaninTetraspanin-30IC50=11
- Tachykinin 3 (Neuromedin K, neurokinin beta), isoform CRA_aTachykinin receptor 3 (NK3)IC50=6
- Epididymis secretory sperm binding proteinHeterogeneous nuclear ribonucleoprotein A1 (hnRNPA1)Kd=1
- PhosphodiesterasePDES1B
- Cyclin-dependent kinase 2, isoform CRA_bCDK2/Bovine cyclin A
- Cyclin-dependent kinase 4, isoform CRA_aCyclin-dependent kinase 4 (CDK 4)
- Kit ligandMast cell growth factorIC50=6
- Dual specificity protein phosphataseMAP kinase phosphatase 3IC50=33
- Phenylalanine hydroxylase, isoform CRA_aPAH
- PCTAIRE protein kinase 2, isoform CRA_aPCTK2Kd=126
- D-amino-acid oxidase isoform 1DAO
- NUAK family, SNF1-like kinase, 1, isoform CRA_aNUAK family SNF1-like kinase 1
- Ubiquitin carboxyl-terminal hydrolaseUbiquitin-specific-processing protease 30IC50=273
- Protein kinase, AMP-activated, beta 1 non-catalytic subunit, isoform CRA_a5''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''''-AMP-activated protein kinase subunit beta-1
- Serine/threonine-protein phosphataseSerine/threonine protein phosphatase PP1-gamma catalytic subunit
- Calcium/calmodulin-dependent protein kinase kinase 2, beta, isoform CRA_fCaM-kinase kinase beta
- Uncharacterized proteinCalcium channel (VER)
- Protein kinase, X-linked, isoform CRA_bSerine/threonine-protein kinase PRKX
- Carbonic anhydraseCarbonic anhydrase V
- Pirin (Iron-binding nuclear protein), isoform CRA_aProbable quercetin 2,3-dioxygenase PIR
- Cadherin 2, type 1, N-cadherin (Neuronal), isoform CRA_bCadherin-2IC50=1
- Aminopeptidasegp150
- Furin (Paired basic amino acid cleaving enzyme), isoform CRA_aHomo sapiens furin (paired basic amino acid cleaving enzyme) (FURIN), mRNA
- Tyrosine-protein kinaseFES
- Aldehyde dehydrogenase 1 family, member A3, isoform CRA_aRetinaldehyde dehydrogenase 3
- TetraspaninTarget of the antiproliferative antibody 1Kd=1
- Discoidin domain receptor family, member 1, isoform CRA_aDiscoidin domain-containing receptor 1 (DDR1)
- VARSValyl-tRNA synthetase 2IC50=3
- EHMT2Histone-lysine N-methyltransferase, H3 lysine-9 specific 3
- Bromodomain containing 2, isoform CRA_bBromodomain and extra-terminal motif (BET)
- Kinesin-like proteinKIFC1IC50=37
- Peroxisome proliferative activated receptor, delta, isoform CRA_aPPAR delta
- Cyclin-dependent kinase inhibitor 1A (P21, Cip1), isoform CRA_aCDK-interacting protein 1IC50=57
- Peptidyl-prolyl cis-trans isomeraseRotamase PPIL1Ki=2
- Mitogen-activated protein kinaseMitogen-activated protein kinase p38
- Mitogen-activated protein kinasep38 MAP kinase alpha/beta
- Non-specific serine/threonine protein kinaseNDR1 protein kinase
- Serine/threonine-protein kinaseProto-oncogene serine/threonine-protein kinase Pim-1
- Vascular endothelial growth factor, isoform CRA_dVPF
- Elongation of very long chain fatty acids protein 5Elongation of very long chain fatty acids protein 5IC50=4
- Nuclear receptor co-repressor 1, isoform CRA_aNuclear receptor corepressor 1
- Intestinal cell (MAK-like) kinase, isoform CRA_aIntestinal cell kinase
- Polymerase (DNA directed), eta, isoform CRA_bDNA polymerase etaIC50=10
- Heat shock protein 90kDa alpha (Cytosolic), class B member 1, isoform CRA_aHeat shock protein HSP 90 (Hsp90)
- Multifunctional fusion proteinMDNCF-a
- C-X-C motif chemokineHSFKd=3
- Alcohol dehydrogenase IB (Class I), beta polypeptide, isoform CRA_aAlcohol dehydrogenase beta chain
- Ubiquitin-conjugating enzyme E2D 3 (UBC4/5 homolog, yeast), isoform CRA_a(E3-independent) E2 ubiquitin-conjugating enzyme D3Kd=5
- PAP2_C domain-containing proteinSGMS2
- HCG18830, isoform CRA_aPHKG1
- Non-specific serine/threonine protein kinaseSerine/threonine-protein kinase LATS2
- High-mobility group box 1, isoform CRA_aHigh mobility group protein 1Kd=9
- HCG30749, isoform CRA_aRB intron encoded G-protein coupled receptorEC50=11
- Retinoblastoma 1 (Including osteosarcoma), isoform CRA_aRbIC50=30
- Epstein-Barr virus induced gene 2 (Lymphocyte-specific G protein-coupled receptor), isoform CRA_aG-protein coupled receptor 183IC50=132
- Carbonic anhydraseβ-Carbonic anhydrase 3 (CA 3)Ki=22
- F420-dependent glucose-6-phosphate dehydrogenaseF420-dependent glucose-6-phosphate dehydrogenase (FGD)Kd=2
- Glycogen synthase kinase-3 beta splice variant X1Tau protein kinase 1 (TPK1)IC50=98
- Cathepsin HCathepsin H
- Cytochrome b562apocytochrome b562(denatured)ITC=2
- DNA gyrase subunit BDNA Gyrase Subunit B
- DNA ligaseDNA ligase
- GlucosylceramidaseGlucosylceramidase precursor (Beta-glucocerebrosidase) (Acid beta-glucosidase) (D-glucosyl-N-acylsphingosine glucohydrolase) (Alglucerase) (Imiglucerase)
- AcetyltransferasePgap1 family proteinEC50=2
- LysR family transcriptional regulatorTranscriptional regulator MvfR
- Diflavin flavoprotein A 3Thioesterase PqsE (PqsE)Kd=2
- Heat shock transcription factor 1 alpha isoformHsf1 proteinEC50=4317
- LysozymeD1.3 mAbITC=44
- Lysozyme GCAM-alpha-lactalbuminITC=6
- Carbonic anhydraseAlpha-carbonic anhydraseKi=37
- Carbonic anhydraseVchβCAKi=35
- Histo-blood group ABO system transferaseGlycoprotein-fucosylgalactoside alpha-N-acetylgalactosaminyltransferase
- Virion spike glycoproteinGP
- Vasoactive intestinal polypeptideVIPKi=218
- Corticotropin releasing hormone receptor 2CRH-R 2
- Peptidylprolyl isomeraseFK506 binding protein 14Ki=1
- Cyclin-dependent kinase 5Cyclin-T1/Cyclin-dependent-like kinase 5
- Amiloride-sensitive cation channel 3Amiloride-sensitive cation channel 3IC50=61
- Adenylate cyclase activating polypeptide 1 (Pituitary) receptor type IPituitary adenylate cyclase-activating polypeptide type I receptor
- Nitric oxide synthaseEndothelial NOS
- Potassium voltage-gated channel, subfamily H (Eag-related), member 2Melanin-concentrating hormone receptor 2/HERG
- Protein kinase, AMP-activated, gamma 2 non-catalytic subunit5'-AMP-activated protein kinase subunit gamma-2EC50=1
- Growth hormone releasing hormone receptorGrowth hormone-releasing hormone receptorIC50=1
- G protein-coupled receptor 154Neuropeptide S receptor
- Ras homolog enriched in brainRHEB2Kd=2
- Beta-lactamaseBeta-lactamaseIC50=1
- Amidases related to nicotinamidaseNicotinamidase (SpNic)Ki=10
- Chloroquine resistance transporterChloroquine resistance transporterIC50=18
- Ubiquitin carboxyl-terminal hydrolaseISOT-3IC50=1
- NS3 protease (Fragment)Protease NS3/Non-structural protein 4A (NS3/NS4A) (D168V)
- NS3 protease (Fragment)Protease NS3/Non-structural protein 4A (NS3/NS4A) (D168V)
- Glucocorticoid receptorNR3C1
- Dihydrofolate reductaseTetrahydrofolate dehydrogenase
- DihydroorotaseDihydroorotase (PyrC)IC50=2
- Kallikrein dThymopsinIC50=21
- Melanocyte-stimulating hormone receptorMC1-R
- Sialidase BSAMEA2203862_00684IC50=5
- 3-oxoacyl-(Acyl carrier protein) synthase IIIPA8380_44470
- Chromosome 1, whole genome shotgun sequenceGlycogen Synthase Kinase 3 (GSK3)IC50=24
- Mobilization protein AMobilization protein AEC50=1
- Serine proteaseGlutamyl endopeptidaseKi=11
- Uncharacterized proteinAldosterone Synthase (CYP11B2)IC50=300
- UDP-N-acetylmuramoyl-L-alanyl-D-glutamate--2,6-diaminopimelate ligaseMurE (E. coli)IC50=3
- Beta-glucuronidaseBeta-glucuronidase (SaGUS)Ki=6
- DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase beta chainIC50=171
- 3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZbeta-Hydroxyacyl-acyl carrier protein dehydratase (FtFabZ)IC50=4
- Cytochrome c oxidase subunit 2Cytochrome c oxidase subunit 2IC50=8
- Edema factorCalmodulin-sensitive adenylate cyclase
- Bifunctional ligase/repressor BirABiotin--[acetyl-CoA-carboxylase] ligaseKi=1
- Cytochrome P450 Cyp144Cytochrome P450 144 (CYP144A1-TRV)Kd=6
- DNA primaseDNA primase (Ba DnaG)IC50=5
- Calmodulin-sensitive adenylate cyclaseCalmodulin-sensitive adenylate cyclase
- Thyroid stimulating hormone beta subunitThyroid-stimulating hormone subunit beta (bTSH)IC50=3
- CAM kinase, CDPK family TgCDPK1Calmodulin-domain protein kinase 1 (CDPK1)IC50=116
- Peptidyl-prolyl cis-trans isomeraseRotamaseKi=2
- Acyl-homoserine lactone acylase PvdQN-terminal nucleophile hydrolase (PVdQ)Ki=4
- Fructose-bisphosphate aldolaseFructose-bisphosphate aldolase, class II
- UDP-N-acetylmuramoyl-tripeptide--D-alanyl-D-alanine ligaseMurF (S. aureus)IC50=1
- SialidasenanI
- Putative hydrolasecifIC50=20
- Diphosphomevalonate decarboxylasediphosphomevalonate decarboxylaseIC50=348
- Mevalonate kinasemevalonate kinaseIC50=953
- Phosphomevalonate kinaseIC50=840
- Plasmepsin VPlasmepsin VIC50=1
- Carbonic anhydrase, family 3Gamma-carbonic anhydraseKi=35
- Inosine-5'-monophosphate dehydrogenaseAB167_18060
- Hypoxanthine phosphoribosyltransferaseHypoxanthine-guanine phosphoribosyltransferase (HGPRT)Ki=23
- Adenylate cyclase type 10AH-related proteinIC50=4
- Epididymis secretory protein Li 18CT2Ki=1
- APOBEC3Aprobable DNA dC->dU-editing enzyme APOBEC-3AIC50=777
- G-protein coupled receptorFree fatty acid receptor 3
- Nonstructural protein NS3-4A (Fragment)Nonstructural protein NS3-4A
- Serine/threonine protein phosphataseSerine/threonine-protein phosphataseKi=11
- Programmed cell death 1 proteinPD1IC50=2
- NeuraminidaseNeuraminidaseIC50=7
- LipoxygenaseSeed linoleate 9S-lipoxygenaseIC50=4
- Amylo-1, 6-glucosidase, 4-alpha-glucanotransferase (Glycogen debranching enzyme, glycogen storage disease type III), isoform CRA_bGlycogen debranching enzymeIC50=23
- Serine/threonine-protein kinase receptor (Fragment)ACVRL1
- Adenosine deaminase isoform 1 (Fragment)Adenosine aminohydrolase
- BCL2-antagonist/killer 1 isoform 1 (Fragment)BCL2L7IC50=13
- G protein-coupled receptor kinase (Fragment)G-protein coupled receptor kinase 2 (GRK2)
- BCL2-like 1 isoform 1 (Fragment)Bcl-2-like protein 1 (Bcl-XL)
- CD40 molecule TNF receptor superfamily member 5 isoform 1 (Fragment)B-cell surface antigen CD40IC50=3
- Ets variant 6 isoform 1 (Fragment)TEL1IC50=1
- Carbonic anhydrase (Fragment)Carbonic anhydrase IX (CA IX)
- Cholesteryl ester transfer protein plasma isoform 1 (Fragment)Lipid transfer protein I
- Cyclin-dependent kinase 7 (MO15 homolog, Xenopus laevis, cdk-activating kinase), isoform CRA_a (Fragment)CDK-activating kinase
- Caspase 2 apoptosis-related cysteine peptidase isoform 1 (Fragment)ICH-1L/1S
- Dopa decarboxylase isoform 1 (Fragment)AADCIC50=15
- Cholesterol side-chain cleavage enzyme, mitochondrial (Fragment)Cholesterol side-chain cleavage enzyme, mitochondrialIC50=1
- Cytochrome b-245 beta polypeptide isoform 1 (Fragment)Heme-binding membrane glycoprotein gp91phox
- Hexosaminidase A isoform 1 (Fragment)Beta-hexosaminidase subunit alpha (HexA)
- Nucleotide diphosphatase (Fragment)NTPaseIC50=1
- Interferon gamma receptor 1 isoform 1 (Fragment)IFN-gamma-R1IC50=2
- Tyrosine-protein kinase (Fragment)2.7.10.2
- Epididymis secretory sperm binding protein (Fragment)Amyloid Binding Alcohol Dehydrogenase
- Myocilin trabecular meshwork inducible glucocorticoid response isoform 1 (Fragment)Myocilin 55 kDa subunitKd=12
- Myeloid/lymphoid or mixed-lineage leukemia translocated to 3 isoform 1 (Fragment)Protein AF-9
- Nucleophosmin isoform 2 (Fragment)NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor)EC50=2
- Phosphodiesterase (Fragment)Phosphodiesterase 9A2
- Protein S100 (Fragment)S-100 protein beta chain
- Serine/threonine-protein phosphatase (Fragment)Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform
- Serine/threonine kinase 11 isoform 1 (Fragment)LKB1
- Growth factor receptor-bound protein 7 isoform 1 (Fragment)Epidermal growth factor receptor GRB-7Kd=31
- Phosphomannomutase (Fragment)phosphomannomutase 2IC50=229
- Protein phosphatase Mg2+/Mn2+ dependent 1D isoform 1 (Fragment)Protein phosphatase 2C isoform delta
- Tyrosine--tRNA ligase (Fragment)Tyrosyl-tRNA synthetase
- Toll-like receptor (Fragment)Toll-like receptor 2
- Phosphodiesterase (Fragment)Phosphodiesterase 9A (PDE9A)
- NCK adaptor protein 1 isoform 1 (Fragment)Nck adaptor protein 1EC50=4
- Receptor-interacting serine-threonine kinase 2 isoform 1 (Fragment)receptor-interacting serine/threonine-protein kinase 2
- Chromobox homolog 4 (Pc class homolog, Drosophila), isoform CRA_a (Fragment)Polycomb 2 homolog
- Vitamin K epoxide reductase complex subunit 1 isoform 1 (Fragment)Vitamin K epoxide reductase complex subunit 1 (hVKORC1)Ki=5
- Ribonuclease P protein componentRNaseP proteinIC50=31
- F420-dependent glucose-6-phosphate dehydrogenaseF420-dependent glucose-6-phosphate dehydrogenase (FGD)Kd=2
- Flavin reductaseNeuraminidase C (NanC)Ki=1
- Integrase (Fragment)Human immunodeficiency virus type 1 integrase
- Integrase (Fragment)HIV-1 IntegraseIC50=129
- Natural resistance-associated macrophage protein 2 isoform 2Natural resistance-associated macrophage protein 2IC50=48
- Dehydrosqualene synthaseDehydrosqualene synthase
- Efflux pump membrane transporterTransporter, hydrophobe/amphiphile efflux-1 (HAE1) familyKd=4
- Testicular tissue protein Li 2C31
- Lysophospholipase II, isoform CRA_fLysophospholipase II
- Methionine aminopeptidase 2Peptidase M 2
- Guanylate cyclaseAtrial natriuretic peptide A-type receptor
- Testicular tissue protein Li 35Cyclin-dependent kinase-like 2Kd=80
- Catechol O-methyltransferaseCatechol O-methyltransferase
- Testicular tissue protein Li 52HSD17B14Ki=49
- DipeptidaseDehydropeptidase-IIC50=33
- Dual specificity phosphatase 23Dual specificity protein phosphatase 23IC50=5
- EPH receptor A3Ephrin type-A receptor 3 (EPHA3)
- Testicular tissue protein Li 73Gamma-glutamyltranspeptidase 1IC50=33
- Glutathione S-transferaseHA subunit 1
- Testicular tissue protein Li 85Serine protease hepsin
- Homeodomain interacting protein kinase 4, isoform CRA_bHomeodomain-interacting protein kinase 4
- Hypoxanthine phosphoribosyltransferaseHGPRTKi=199
- Delta-aminolevulinic acid dehydrataseALADH
- Testicular tissue protein Li 96GAPB3
- cGMP-dependent protein kinasecGMP-dependent protein kinase 2
- Testicular tissue protein Li 130Ornithine delta-aminotransferaseKi=2
- Testicular tissue protein Li 135Proprotein convertase PC4Ki=6
- PhosphodiesterasecAMP-specific 3',5'-cyclic phosphodiesterase 4D
- Testicular tissue protein Li 138Xaa-Pro dipeptidase
- Proteasome subunit beta20S proteasome
- Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit BSerine/threonine protein phosphatase 2A, 55 kDa regulatory subunit B, alpha isoformIC50=1
- Superoxide dismutase [Cu-Zn]EC-SODIC50=4
- Serine/threonine kinase 32C, isoform CRA_dSerine/threonine-protein kinase 32C
- Testicular tissue protein Li 188STK36Kd=136
- Testicular tissue protein Li 209Heat shock protein 75 kDa, mitochondrial
- Ubiquitin carboxyl-terminal hydrolaseUbiquitin carboxyl-terminal hydrolase 5
- Ubiquitin carboxyl-terminal hydrolaseUbiquitin C-terminal Hydrolase L3 (UCH-L3)
- Testicular secretory protein Li 13Carnitine O-palmitoyltransferase 2, mitochondrial
- Testicular secretory protein Li 24Lecithin-cholesterol acyltransferase (LCAT)IC50=4
- Leukotriene A(4) hydrolaseLeukotriene A-4 hydrolase (LTA4H)
- Testicular secretory protein Li 28Serine/threonine-protein kinase MAKKd=79
- Protein phosphatase methylesterase 1protein phosphatase methylesterase 1IC50=5
- Proteasome subunit alpha typePSMA6EC50=14
- Proteasome subunit betaProteasome component C5
- Testicular secretory protein Li 54STAM-binding protein (AMSH)IC50=28
- Testicular secretory protein Li 59HBV XAg-transactivated protein 3IC50=5
- Testicular secretory protein Li 64UBA domain-containing protein 1Ki=13
- Vacuolar proton pump subunit BV-type proton ATPase subunit B, brain isoformIC50=1
- Aspartate aminotransferasecCATIC50=93
- Adenylate kinase 2, mitochondrialAdenylate kinase 2, mitochondrialKi=4
- Testis secretory sperm-binding protein Li 224nPCTK1
- Testis secretory sperm-binding protein Li 236PDihydropteridine reductaseKi=1
- Glutathione S-transferase A2HA subunit 2IC50=33
- Kinesin-like proteinKinesin-like protein KIF2CIC50=1
- Testis tissue sperm-binding protein Li 69n26S Proteasome regulatory subunit Rpn11 (Rpn11)IC50=516
- G-protein coupled receptor 139GPR139
- Major capsid protein L1L1
- Beta-lactamaseMetallothioprotein beta-lactamase IIIC50=59
- Broad-substrate range phospholipase CPLC
- PHD finger protein SPOC1SPOC1IC50=1
- Alpha-glucosidaseAlpha-xylosidaseIC50=3
- Pyrroline-5-carboxylate reductaseP5CR
- ETO24.4.1.14
- AGD2DAPIC50=60
- DXS1DXSIC50=5
- FAC1AtAMPDIC50=1
- Peptide deformylasePeptide deformylase 1A, chloroplasticIC50=24
- HK3Histidine kinaseEC50=16
- Signal peptidase ISignal peptidase IBIC50=1
- Beta-lactamaseblaIC50=16
- Lipoprotein lipaseLPLIC50=73
- PhosphodiesterasePhosphodiesterase 10 (PDE10)
- BMA-GOB-1Trehalose-6-phosphate phosphataseKi=9
- Genome polyprotein3D polymeraseKi=26
- Uncharacterized proteinLOAG_11860Ki=1
- Type III pantothenate kinase2.7.1.33Ki=1
- MyoglobinMBIC50=4
- Orf1a proteinGrowth factor-like peptide
- RAR related orphan receptor B isoform 2Nuclear receptor ROR-beta
- Attachment glycoproteinGlycoprotein GEC50=7
- Polypeptide N-acetylgalactosaminyltransferaseUDP-GalNAc:polypeptide N-acetylgalactosaminyltransferase 2IC50=2
- Uncharacterized proteinbeta-actinIC50=4
- Protein kinase domain-containing proteinXAIRK2-AIC50=3
- Quorum-sensing regulator protein FQuorum-sensing regulator protein FIC50=3
- Kallikrein 1, renal/pancreas/salivary, isoform CRA_aKallikrein-1 (KLK1)
- Kallikrein LKallikrein-13
- NH(3)-dependent NAD(+) synthetaseBAS1855IC50=124
- Adenosine deaminaseAdenosine deaminase 3 (SanADA3)Ki=2
- Pregnancy-associated glycoproteinPepsinIC50=5
- S9 family peptidaseProlyl endopeptidase
- alpha-1B adrenergic receptorADRA1BKi=117
- Major prion proteinPRP
- 3-hydroxy-3-methylglutaryl coenzyme A reductaseHMG-CoA reductaseIC50=15
- chymaseChymaseIC50=309
- Uncharacterized proteinUncharacterized proteinKi=1
- ABHD16AProtein BAT5IC50=2
- AGERRAGE
- CFBComplement factor BIC50=283
- GABBR1Gb1
- Proteasome subunit betaRING12IC50=59
- NOTCH4INT3IC50=1
- MDC1Mediator of DNA damage checkpoint protein 1IC50=7
- Cytochrome c oxidase subunit 2Cytochrome c oxidase subunit 2IC50=16
- Cytochrome c oxidase subunit 1Cytochrome c oxidase subunit 1IC50=2
- NADH-ubiquinone oxidoreductase chain 4Mitochondrial complex I (NADH dehydrogenase)IC50=5
- HTH-type transcriptional regulator TtgRTranscriptional Regulator TtgR Mutant R176GITC=2
- Beta-lactamaseMetallo-beta-lactamase superfamily protein
- Beta-lactamase3.5.2.6Ki=4
- Glyco_18 domain-containing proteinChitinase B1
- NOL1/NOP2/sun family proteinBeta-xylosidaseKi=1
- Alpha-galactosidaseAlpha-galactosidase CIC50=1
- Opioid receptor delta 1G_PROTEIN_RECEP_F1_2 domain-containing protein
- Probable nicotinate-nucleotide adenylyltransferaseNicotinic acid mononucleotide adenylyltransferase (NaMNAT)
- Protein E6 (Fragment)Protein E6IC50=4
- Protein E6 (Fragment)Protein E6IC50=4
- Protein E6 (Fragment)Protein E6IC50=4
- 5-hydroxytryptamine receptor 4 transcript variant b2HTR4
- Epoxide hydrolase 1Epoxide hydrolase 1IC50=14
- Glutamate racemaseGlutamate racemaseKi=4
- G-protein coupled receptor 119G-protein coupled receptor 119EC50=1
- Gonadotropin releasing hormone receptorGonadotropin releasing hormone receptor (GNRHR)IC50=2
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunitPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/gamma isoform
- Replicative DNA helicasednaBIC50=30
- ATP-binding cassette subfamily B member 11Abcb11
- Rho-associated protein kinaseRho-associated protein kinase 2 (ROCK-2)
- Toxin ParEparEIC50=57
- Rhomboid family intramembrane serine proteaseRhomboid protease (HiGlpG)IC50=3
- DNA primase TraCDNA primase traCIC50=1
- DNA gyrase subunit BDNA gyrase subunit B (DNA gyraseB)IC50=51
- DNA topoisomerasesupXIC50=22
- Glyceraldehyde-3-phosphate dehydrogenaseGlyceraldehyde-3-phosphate dehydrogenase, glycosomal
- Bifunctional dihydrofolate reductase-thymidylate synthaseBifunctional dihydrofolate reductase-thymidylate synthase
- Putative trypanothione reductaseTR
- PIK3R1 (Fragment)Phosphoinositide 3-Kinase (PI3K) Chain B
- CHN2 (Fragment)Rho-GTPase-activating protein 3Ki=1
- Lethal factorAnthrax Lethal Factor (LF)
- Indoleamine 2,3-dioxygenase 1IDO
- 4-diphosphocytidyl-2-C-methyl-D-erythritol kinaseCMKIC50=6
- Enoyl-[acyl-carrier-protein] reductase [NADH]Enoyl-ACP reductase (Wt ypFabV)
- Fructose-bisphosphate aldolaseFructose-bisphosphate aldolase, class II
- T3SS effector protein kinase YopO/YpkAProtein kinase AIC50=4
- Regulatory protein E2Human papillomavirus regulatory protein E2Kd=38
- DNA topoisomerase 1supXIC50=22
- Protein E6Protein E6IC50=4
- Protective antigenProtective antigenEC50=8
- Dihydropteroate synthaseDihydropteroate synthase
- Protein-L-isoaspartate O-methyltransferaseProtein-beta-aspartate methyltransferaseKi=8
- Epididymis secretory sperm binding proteinTyrosyl-DNA phosphodiesterase 2
- Thymidine kinaseThymidine kinase, cytosolic
- Ribosomal protein S6 kinasep90-RSK 3
- Epididymis secretory sperm binding proteinFatty acid binding protein muscle
- Epididymis secretory sperm binding proteinguanine nucleotide-binding protein subunit alpha-15
- S-methyl-5'-thioadenosine phosphorylaseMethylthioadenosine Phosphorylase (MTAP)
- Epididymis secretory sperm binding proteinNT5CPKi=6
- FascinHSNIC50=31
- Epididymis secretory sperm binding proteinICAM-1IC50=213
- Epididymis secretory sperm binding proteinV-ATPase S1 accessory proteinIC50=12
- Epididymis secretory sperm binding proteinSerine/threonine-protein kinase 3 (MST2)
- GalectinPutative MAPK-activating protein PM12
- Phosphate transporterGLVR-2IC50=12
- Epididymis secretory sperm binding proteinLysine-specific demethylase 5D (KDM5D)IC50=6
- Phosphoinositide phospholipase CPhospholipase C-delta-1Kd=1
- m7GpppX diphosphataseScavenger mRNA-decapping enzyme (DcpS)
- AdenosylhomocysteinaseAdenosylhomocysteinase
- RuvB-like helicasePontin 52IC50=2
- Epididymis secretory sperm binding proteinGLP2REC50=88
- Epididymis secretory sperm binding proteinCell division cycle 7-related protein kinase
- EPH receptor A5, isoform CRA_aEphrin type-A receptor 5
- Signal transducer and activator of transcriptionTranscription factor STAT5a (STAT5a)
- Inosine-5'-monophosphate dehydrogenaseInosine-5 -monophosphate dehydrogenase 2
- SulfurtransferaseThiosulfate sulfurtransferaseIC50=62
- Glucose-6-phosphate 1-dehydrogenaseglucose-6-phosphate 1-dehydrogenase isoform b
- UDP-glucose 4-epimeraseUDP-glucose 4-epimeraseIC50=6
- Epididymis secretory sperm binding proteinCarbonyl reductase [NADPH] 1
- Epididymis secretory sperm binding proteinDual specificity protein phosphatase 22
- Aldehyde dehydrogenase 2 family (Mitochondrial), isoform CRA_cAldehyde dehydrogenase (ALDH2)
- Epididymis secretory sperm binding proteinProtein kinase C-interacting protein 1
- Epididymis secretory sperm binding proteinSpermidine/spermine N(1)-acetyltransferase 1
- Epididymis secretory sperm binding proteinNon-specific lipid-transfer proteinKd=2
- Epididymis secretory sperm binding proteinPlatelet-derived growth factor subunit B (PDGFB)
- Glutathione S-transferaseGSTM2-2
- Epididymis secretory sperm binding proteinH-PGDS
- CatalaseCATIC50=4
- Adenylate cyclaseAdenylate cyclase
- Cannabinoid receptor 1CB1
- Serine proteaseSerine protease SplBKi=12
- Bifunctional ligase/repressor BirABiotin protein ligase (BPL)
- Peptide deformylasePeptide deformylaseIC50=54
- Alpha-galactosidaserafAIC50=1
- ChitinaseChitinase B
- Carbonic anhydraseCAMKi=112
- HMWP2 nonribosomal peptide synthetaseirp2
- Acetyltransferase, GNAT familyEis_Ban acetyltransferase (Eis_Ban)IC50=3
- Malate dehydrogenaseMalate dehydrogenaseIC50=21
- PhospholipasePhospholipase D (PldA)IC50=32
- Pol protein (Fragment)HIV-1 IntegraseIC50=129
- HAD super, subIIIB family proteinAcid phosphatase (acpB)Ki=8
- Enoyl-[acyl-carrier-protein] reductase [NADH]Enoyl-[acyl-carrier-protein] reductase [NADH]
- Chymotrypsin-like elastase family member 1Elastase
- DipeptidaseRenal dipeptidaseKi=188
- Malate dehydrogenaseMDH1
- Dipeptidyl peptidase 4Dipeptidyl peptidase IV soluble form
- Calpain small subunit 1 isoform 1Calcium-dependent protease small subunit 1Ki=27
- Prolyl endopeptidasePE
- ArylsulfataseASIC50=2
- MHC class II antigenHuman leukocyte antigen DR beta chainIC50=27
- Zinc metalloproteinaseZinc metalloproteinase dpy-31IC50=5
- Trehalose-6-phosphate synthase, putativeTrehalose-6-phosphate phosphataseKi=9
- Sialidase B (Neuraminidase B)Neuraminidase B (NanB)
- Modulator of drug activity AModulator of drug activity AIC50=17
- DNA-directed RNA polymerase subunit betaDNA-directed RNA polymerase beta chainIC50=45
- Methionine aminopeptidaseMethionine Aminopeptidase (MAP)IC50=393
- Thiol:disulfide interchange proteinJW3832Kd=21
- Glyoxylate bypass operon transcriptional repressor IclRAcetate Operon Repressor (IclR)ITC=4
- S-ribosylhomocysteine lyaseS-ribosylhomocysteine lyaseKi=3
- Phosphopantetheine adenylyltransferaseDephospho-CoA pyrophosphorylaseIC50=28
- Glutamine synthetaseGlutamine synthetase
- 5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase (MTAN)
- Beta sliding clampJW3678
- Tyrosine--tRNA ligaseTyrosine--tRNA ligaseKi=2
- HTH-type transcriptional repressor AllRNegative regulator of allantoin and glyoxylate utilization operonsITC=1
- D-alanine--D-alanine ligaseD-alanylalanine synthetase BIC50=2
- Biotin carboxylaseBiotin CarboxylaseIC50=14
- Carbamoyl-phosphate synthase small chainCarbamoyl-phosphate synthetase
- Fructose-bisphosphate aldolaseFructose-bisphosphate aldolase class 2Ki=6
- Chaperone SurAsurAIC50=5
- Inosine-5'-monophosphate dehydrogenaseInosine-5-monophosphate dehydrogenase (IMPDH)IC50=9
- Glucose-1-phosphate cytidylyltransferaseCDP-glucose pyrophosphorylaseKi=1
- Cysteine proteinase exotoxin SpeBCysteine protease SpeB (SpeB)
- CollagenaseGelatinase ColGIC50=3
- Alanine racemaseAlanine racemaseKi=8
- Methionine aminopeptidaseMethionine Aminopeptidase (MAP)IC50=393
- 4-hydroxy-3-methylbut-2-enyl diphosphate reductaseLytBKi=1
- Endoribonuclease MazFmRNA interferase toxin, antitoxin is MazEEC50=948
- TrehalaseTrehalaseIC50=10
- G_PROTEIN_RECEP_F1_2 domain-containing proteinDOPAMINE D2Ki=28
- Protein kinase domain-containing proteinCSNK1DIC50=29
- Uncharacterized proteinGABA A BenzodiazepineKi=10
- Uncharacterized proteinArachidonate 5-lipoxygenaseIC50=1
- G_PROTEIN_RECEP_F1_2 domain-containing proteinNPY-Y4Ki=11
- G_PROTEIN_RECEP_F1_2 domain-containing proteinHTR6Ki=3
- Hydroxycarboxylic acid receptor 1Hydroxycarboxylic acid receptor 1EC50=1
- Hydroxycarboxylic acid receptor 1Hydroxycarboxylic acid receptor 1EC50=17
- Hydroxycarboxylic acid receptor 2G-protein coupled receptor HM74A
- Dihydrofolate reductasebaDHFR
- Beta-lactamaseβ-lactamase (Bla2)
- DNA primaseDNA primase (Ba DnaG)IC50=5
- Inosine-5'-monophosphate dehydrogenaseAB167_18060
- Replicative DNA helicasednaBIC50=30
- CD4T-cell surface antigen T4/Leu-3
- Regulatory protein E2Regulatory protein E2Kd=1
- Polysaccharide deacetylase family proteinPeptidoglycan GlcNAc deacetylase
- Dihydrofolate reductaseTetrahydrofolate dehydrogenaseIC50=27
- Polysaccharide deacetylasePeptidoglycan GlcNAc deacetylase
- Bifunctional cytochrome P450/NADPH--P450 reductaseCytochrome P450 monooxygenase BM3 (BM3)Kd=1
- DNA repair and recombination protein RadADNA repair and recombination protein (RadA)Kd=8
- Type-2 restriction enzyme BamHIType-2 restriction enzyme BamHIIC50=4
- Kynurenine 3-monooxygenaseKynurenine 3-monooxygenaseIC50=2
- Epoxide hydrolaseEpoxide hydrolaseIC50=16
- Muscarinic acetylcholine receptorCHRM4Ki=27
- Potassium voltage-gated channel subfamily J member 5CIR
- Thioredoxin reductaseThioredoxin reductaseKi=18
- Trypanothione_reductaseTrypanothione reductaseIC50=64
- NAD-dependent protein deacetylaseSIR2-like proteinIC50=21
- Sterol_14-alpha-demethylase_-_putativeSterol 14α-demethylase (CYP51)Kd=7
- Threonine--tRNA ligasey1903Ki=24
- T3SS effector protein-tyrosine-phosphatase YopHSecreted effector protein
- Thymidine phosphorylaseThymidine phosphorylase (TP)IC50=11
- Zinc metalloproteinaseZinc metalloproteinase dpy-31IC50=5
- 4-hydroxyphenylpyruvate dioxygenase4-hydroxyphenylpyruvic acid oxidase
- DNA topoisomerase (ATP-hydrolyzing)DNA gyrase subunit BIC50=352
- Phospholipase DPLD alpha C2 domainITC=1
- 2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthaseMDSIC50=1
- Isoleucine--tRNA ligaseIleRSIC50=37
- Arachidonate 15-lipoxygenase15-Lipoxygenase (LoxA)IC50=15
- Orf1ab polyproteinORF1ab polyprotein
- SHORT (C15) CHAIN Z-ISOPRENYL DIPHOSPHATE SYNTHASE (Z-FPP SYNTHASE) (Z-FARNESYL DIPHOSPHATE SYNTHASE) (Z-FPP SYNTHETASE) (Z-FARNESYL DIPHOSPHATE SYNTHETASE) (GERANYLTRANSTRANSFERASE) (FARNESYL PYROPHOSPHATE SYNTHETASE)cis-Farnesyl diphosphate synthase (cis-FPPS)IC50=8
- MAL32 isoform 1 (Fragment)Alpha-glucosidase MAL32IC50=11
- NCE103 isoform 1 (Fragment)β-Carbonic anhydrase (CA)Ki=14
- Botulinum neurotoxin type BBotulinum neurotoxin B light chainIC50=2
- ORF1ab polyproteinORF1ab polyprotein
- Heme-binding protein AGlutathione-binding protein (GbpAPm)Kd=3
- Transcription termination factor RhoRho Transcription Termination FactorITC=3
- Beta-ketoacyl-ACP synthase I3-oxoacyl-[acyl-carrier-protein] synthase 1IC50=40
- Disulfide bond formation protein DsbBDisulfide oxidoreductaseIC50=8
- UDP-N-acetylglucosamine 1-carboxyvinyltransferaseEPT
- Xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferase (XGPRT)Ki=2
- Recombinase RecAProtein RecA
- Cystathionine beta-lyaseCBLIC50=23
- Peptide deformylasePolypeptide deformylase
- ATP-dependent Clp endopeptidase proteolytic subunit ClpPATP-dependent Clp protease proteolytic subunitKd=2
- DNA-directed RNA polymerase subunit betaJW3951IC50=4
- Type 3 dihydrofolate reductaseBacterial dihydrofolate reductase
- Acyl-ACP--UDP-N-acetylglucosamine O-acyltransferaseUDP-N-acetylglucosamine acryltransferase (LpxA)Kd=8
- Inorganic diphosphataseInorganic pyrophosphatase (EcPPiase)IC50=14
- TryptophanaseL-tryptophan indole-lyaseKi=4
- DNA polymerase IDNA polymerase IIC50=4
- UDP-3-O-acyl-N-acetylglucosamine deacetylaseUDP-3-O-[3-hydroxymyristoyl] N-acetylglucosamine deacetylase (LxpC)
- Thymidylate synthaseTS
- Serine--tRNA ligase6.1.1.11Ki=2
- Ribonuclease HIRibonuclease HIC50=18
- (2E,6E)-farnesyl diphosphate synthaseFPP synthaseIC50=5
- Nicotinate-nucleotide adenylyltransferaseNicotinate mononucleotide adenylyltransferase (NadD)
- Uracil phosphoribosyltransferaseuraPKi=1
- DNA topoisomeraseDNA topoisomeraseIC50=4
- Niemann-Pick C1-like 1 proteinNiemann-Pick C1-like 1 proteinIC50=4
- Niemann-Pick C1-like 1 proteinNiemann-Pick C1-like 1 proteinIC50=4
- Chemokine (C-X-C motif) receptor 6CXCR-6
- Chemokine (C-C motif) receptor 7C-C chemokine receptor type 7
- Chemokine (C-C motif) receptor 4C-C chemokine receptor type 4 (CCR4)
- C-C motif chemokineMacrophage inflammatory protein 1-alphaIC50=7
- Burkitt lymphoma receptor 1, GTP binding protein (Chemokine (C-X-C motif) receptor 5)C-X-C chemokine receptor type 5
- Cytochrome P450, family 1, subfamily A, polypeptide 1P450-P1
- A-glucosidaseAlpha-glucosidaseIC50=6
- Enoyl-[acyl-carrier-protein] reductase [NADH]fablKi=20
- Calcium dependent protein kinaseCalcium dependent protein kinaseIC50=1
- Testis tissue sperm-binding protein Li 55eTestis-specific serine/threonine-protein kinase 1
- HCG1641087Testis-specific serine/threonine-protein kinase 2
- Beta-lactamaseBeta-lactamaseIC50=2
- Beta-lactamaseBeta-lactamase SCO-1IC50=3
- D-alanyl-D-alanine dipeptidaseD-Ala-D-Ala dipeptidase
- CCAP-like receptorNeuropeptide S receptor
- TANK-binding kinase 1TANK-binding kinase 1IC50=23
- Glutamate metabotropic receptor 4metabotropic glutamate 4
- Chemokine binding protein 2, isoform CRA_aD6
- Chemokine (C-C motif) receptor 3, isoform CRA_aC-C chemokine receptor type 3
- Parathyroid hormone receptor 1, isoform CRA_aPTH1 receptor
- Ubiquitin carboxyl-terminal hydrolaseUbiquitin carboxyl-terminal hydrolase 4IC50=1
- Ubiquitin-activating enzyme E1-like 2, isoform CRA_aMOP-4IC50=17
- ATP-binding cassette, sub-family G (WHITE), member 2, isoform CRA_aBCRP
- Elongation of very long chain fatty acids protein 6Elongation of very long chain fatty acids protein 6IC50=132
- EPH receptor A4, isoform CRA_aEphrin type-A receptor 4
- Protein tyrosine phosphatase, non-receptor type 7, isoform CRA_aTyrosine-protein phosphatase non-receptor type 7 (HEPTP)
- Choline/ethanolamine phosphotransferase 1, isoform CRA_bhCEPT1IC50=45
- Endothelin converting enzyme 1, isoform CRA_bEndothelin-converting enzyme 1 (ECE1)
- Cytochrome P450 14alpha-demethylaseCytochrome P450 14alpha-demethylaseKd=31
- Angiotensin-converting enzymeAngiotensin-Converting EnzymeIC50=6
- Mast cell-restricted serine protease 7Tryptase alpha/beta-1Ki=3
- BCR/ABL p210 fusion protein (Fragment)fusionEC50=1
- Carboxylic ester hydrolaseCG8425-PA [Drosophila melanogaster]IC50=21
- Ntsr1 proteinNeurotensin receptor 1
- G protein-coupled receptor 142Gpr142
- Opioid receptor, delta 1Delta-type opioid receptor
- Retinoid X receptor alphaRetinoid X receptor alpha
- Calcitonin receptor-likeCrlrKi=1
- Rapgef4 proteincAMP-dependent Rap1 guanine-nucleotide exchange factorIC50=50
- Arachidonate 12-lipoxygenaseArachidonate 12-lipoxygenaseIC50=29
- Arachidonate 15-lipoxygenaseArachidonate 15-lipoxygenaseIC50=3
- Clan CD, family C13, asparaginyl endopeptidase-like cysteine peptidaseAsparaginyl Endopeptidase (AE)IC50=30
- Cryptochrome 2 (Photolyase-like), isoform CRA_aCryptochrome-2EC50=54
- Beta-lactamasePER-2 beta-lactamase
- PhosphodiesterasecAMP-specific 3',5'-cyclic phosphodiesterase 4DIC50=15
- Legumainasparaginyl endopeptidaseIC50=19
- Phosphatidylinositol-4-phosphate 3-kinase, catalytic subunit type 2 betaPIK3C2B
- Putative lanosterol 14-alpha-demethylaseSterol 14α-demethylase (CYP51)Kd=7
- Vasopressin V1a receptorAVPR1AKi=2
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)Hepatitis C virus NS3 protease/helicase
- Genome polyprotein (Fragment)NS3IC50=146
- Beta-lactamaseblaSHV-95Ki=4
- Cell division control protein 28, putativeCell division control protein 28, putativeIC50=1
- Calmodulin-domain protein kinase 1, putativeCalmodulin-domain protein kinase 1, putativeIC50=133
- Mitogen-activated protein kinaseMitogen-activated protein kinaseIC50=1
- Fanconi anemia, complementation group FFanconi anemia group F proteinKd=1
- Beta-glucuronidaseEnsembl:ENSBTAP00000000941IC50=217
- TGF-beta receptor type-2TGF-beta receptor type II
- Carboxylic ester hydrolase (Fragment)3.1.1.-IC50=2
- ATP-dependent RNA helicase DDX1DEAD box protein retinoblastomaIC50=7
- Thymidine kinaseThymidine kinaseIC50=17
- Neuropeptide YNeuropeptide YKi=5
- Chromobox homolog 3 (HP1 gamma homolog, Drosophila)Modifier 2 proteinKd=1
- CD36 antigen (Collagen type I receptor, thrombospondin receptor)FATIC50=6
- Glutamate metabotropic receptor 3metabotropic glutamate 3
- ATP-binding cassette, sub-family B (MDR/TAP), member 1Multidrug resistance protein 1/Multidrug resistance associated protein 1
- Protein-serine/threonine kinasePyruvate dehydrogenase kinase isoform 4
- Muscarinic acetylcholine receptorRecName: Full=Muscarinic acetylcholine receptor M2
- Poly (ADP-ribose) polymerase family, member 12, isoform CRA_bZinc finger CCCH domain-containing protein 1IC50=21
- Calcium/calmodulin-dependent protein kinase (CaM kinase) II betaCaM kinase II beta
- Receptor (Calcitonin) activity modifying protein 3RAMP3Ki=1
- 5-hydroxytryptamine (Serotonin) receptor 5A5-hydroxytryptamine receptor 5A
- Ras-related C3 botulinum toxin substrate 1 (Rho family, small GTP binding protein Rac1)Rac1 proteinIC50=21
- Erythromycin ribosome methylaserRNA adenine N-6-methyltransferaseKi=31
- ACBD3 protein (Fragment)Benzodiazepine centralKi=1
- GRIK1 proteinGRIK1 proteinKi=1
- Galectin-3Galectin-3IC50=18
- Trypanothione reductaseTrypanothione reductaseIC50=64
- Beta-lactamaseGil1IC50=2
- Mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 1 (MEK)
- Cereblon isoform 4Cereblon isoform 4
- NeuraminidaseNeuraminidase N1IC50=2
- Beta-galactosidaseBeta-galactosidaseIC50=5
- Beta-lactamaseBeta-lactamase ACC-4IC50=6
- Motilin receptorMotilin receptor
- ATP-binding cassette, sub-family C (CFTR/MRP), member 1Multidrug resistance-associated protein 1
- HRH1 proteinHRH1 proteinKi=2
- Histone deacetylase 8Histone deacetylase 8
- Purinergic receptor P2Y G-protein coupled 14 transcript variant 2Insulin Receptor-Related Protein (INSRR)
- Dihydroorotate dehydrogenase, mitochondrial, putativeDihydroorotate Dehydrogenase (DHODH)IC50=11
- Orotidine 5' monophosphate decarboxylase, putativeODCaseKi=2
- KCNH2 proteinKCNH2 proteinKi=1
- Cell division protein FtsZCell division protein FtsZIC50=1
- NeuraminidaseNeuraminidase