WIPO

Data

Cmpds

HGNC*

WIPO Title

Organization

Deposition

Downloads

110

3-AMINO PYRROLIDINE AND PIPERIDINE MACROCYCLIC OREXIN RECEPTOR AGONISTS

MERCK SHARP & DOHME LLC

10/05/22

2D 3D TSV

32

POLYHETEROCYCLIC GLP-1 R MODULATING COMPOUNDS

GILEAD SCIENCES, INC.

10/05/22

2D 3D TSV

31

SARS-COV-2 MPRO INHIBITOR COMPOUNDS

HEPTARES THERAPEUTICS LIMITED

10/05/22

2D 3D TSV

49

1-(2-(4-CYCLOPROPYL-1H-1,2,3-TRIAZOL-1-YL)ACETYL)-4-HYDROXY-N-(BENZYL)PYRROLIDIN E-2-CARBOXAMIDE DERIVATIVES AS VHL INHIBITORS FOR THE TREATMENT OF ANEMIA AND CANCER

GENENTECH, INC.

08/07/22

2D 3D TSV

42

1-(2-(4-CYCLOPROPYL-1H-1,2,3-TRIAZOL-1-YL)ACETYL)-4-HYDROXYPYRROLIDINE-2-CARBOXA|MIDE DERIVATIVES AS VHL INHIBITORS FOR THE TREATMENT OF ANEMIA

GENENTECH, INC.

08/07/22

2D 3D TSV

56

7-AZOLE SUBSTITUTED 2-AMINOQUINAZOLINE INHIBITORS OF HPK1

MERCK SHARP & DOHME LLC

08/07/22

2D 3D TSV

80

CYCLOPENTATHIOPHENE CARBOXAMIDE DERIVATIVES AS PLATELET ACTIVATING FACTOR RECEPTOR ANTAGONISTS

BOEHRINGER INGELHEIM INTERNATIONAL GMBH

08/07/22

2D 3D TSV

47

DIAMINOPYRIMIDINE CARBOXAMIDE INHIBITORS OF HPK1

MERCK SHARP & DOHME LLC

08/07/22

2D 3D TSV

14

N-[2-({4-[3-(ANILINO)-4-OXO-4,5,6,7-TETRAHYDRO-1H-PYRROLO[3,2-C]PYRIDIN-2-YL]PYRIDIN-3-YL)OXY)ETHYL]PROP-2-ENAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER

BAYER AKTIENGESELLSCHAFT

08/07/22

2D 3D TSV

34

PYRAZOLE DERIVATIVES ASR ET KINASE INHIBITORS

ELI LILLY AND COMPANY

08/07/22

2D 3D TSV

125

SMALL MOLECULE INHIBITORS OF NF-KB INDUCING KINASE

JANSSEN PHARMACEUTICA NV

08/07/22

2D 3D TSV

384

7-PHENYL SUBSTITUTED 2-AMINOQUINAZOLINE INHIBITORS OF HPK1

MERCK SHARP & DOHME LLC

07/22/22

2D 3D TSV

61

HETEROCYCLIC SPIRO COMPOUNDS AND METHODS OF USE

AMGEN INC.

07/21/22

2D 3D TSV

226

INTERLEUKIN-17 INHIBITORS

NOVARTIS AG

07/21/22

2D 3D TSV

236

N-LINKED ISOQUINOLINE AMIDES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF

MERCK SHARP & DOHME LLC

07/21/22

2D 3D TSV

219

SUBSTITUTED 1H-PYRAZOLO[4,3-C]PYRIDINES AND DERIVATIVES AS EGFR INHIBITORS

BOEHRINGER INGELHEIM INTERNATIONAL GMBH

07/21/22

2D 3D TSV

68

SUBSTITUTED MORPHOLINE COMPOUNDS

GENENTECH, INC.

07/21/22

2D 3D TSV

19

ANTIVIRAL HETEROARYL KETONE DERIVATIVES

PFIZER INC.

06/09/22

2D 3D TSV

80

NOVEL CORONAVIRUS MAIN PROTEASE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

SICHUAN UNIVERSITY

06/09/22

2D 3D TSV

29

COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CRYPTOSPORIDIOSIS

NOVARTIS AG

05/24/22

2D 3D TSV

71

PHOSPHOLIPID COMPOUNDS AND USES THEREOF

GILEAD SCIENCES, INC.

05/24/22

2D 3D TSV

229

SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER

THE BROAD INSTITUTE, INC.

05/24/22

2D 3D TSV

68

SUBSTITUTED ACYL SULFONAMIDES FOR TREATING CANCER

THE BROAD INSTITUTE, INC.

05/24/22

2D 3D TSV

294

TRIAZOLOPYRIDINYL COMPOUNDS AS KINASE INHIBITORS

BRISTOL-MYERS SQUIBB COMPANY

05/24/22

2D 3D TSV

83

HGNC:3827 3826

AMINOIMIDAZOLE FPR2 AGONISTS

BRISTOL-MYERS SQUIBB COMPANY

05/02/22

2D 3D TSV

172

CYCLIN-DEPENDENT KINASE 7 (CDK7) NON-COVALENT INHIBITORS

JANSSEN PHARMACEUTICA NV

05/02/22

2D 3D TSV

25

DIHYDROOROTATE DEHYDROGENASE INHIBITORS

JANSSEN BIOTECH, INC.

05/02/22

2D 3D TSV

6

DIHYDROOROTATE DEHYDROGENASE INHIBITORS

JANSSEN BIOTECH, INC.

05/02/22

2D 3D TSV

8

DIHYDROOROTATE DEHYDROGENASE INHIBITORS

JANSSEN BIOTECH, INC.

05/02/22

2D 3D TSV

141

PREPARATION OF BENZIMIDAZOLONE DERIVATIVES AS NOVEL DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 INHIBITORS

MERCK SHARP & DOHME CORP.

05/02/22

2D 3D TSV

168

PREPARATION OF OXINDOLE DERIVATIVES AS NOVEL DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 INHIBITORS

MERCK SHARP & DOHME CORP.

05/02/22

2D 3D TSV

100

Aminocarbamoyl compounds for the treatment of viral infections

F. Hoffmann-La Roche Ag

03/30/22

2D 3D TSV

178

Sars-cov-2 inhibitors having covalent modifications for treating coronavirus infections

Insilico Medicine Ip Limited

01/27/22

2D 3D TSV

44

Compounds and method of treating covid-19

Pfizer Inc.

01/13/22

2D 3D TSV

3

Compounds and methods for the treatment of covid-19

Pfizer Inc.

01/13/22

2D 3D TSV

94

Nitrile-containing antiviral compounds

Pfizer Inc.

01/13/22

2D 3D TSV

12

Anticoronaviral compounds and compositions, their pharmaceutical uses and materials for their synthesis

Pfizer Inc.

01/31/21

2D 3D TSV

61

Anticoronviral compounds and compositions, their pharmaceutical uses and materials for their synthesis

Pfizer Inc.

10/17/20

2D 3D TSV