Target Name
Affinity Link(s)
Article(s)
UniProt
Files
1D-myo-inositol 2-acetamido-2-deoxy-alpha-D-glucopyranoside deacetylase
Ki: 3 IC50: 6
2
2D 3D TSV 
5'-AMP-activated protein kinase subunit beta-2
EC50: 10
4
2D 3D TSV 
5'-AMP-activated protein kinase subunit gamma-1
IC50: 1 EC50: 10
5
2D 3D TSV 
85/88 kDa calcium-independent phospholipase A2
IC50: 63
3
2D 3D TSV 
Abscisic acid receptor PYL1/Protein phosphatase 2C 16
IC50: 10
1
2D 3D TSV 
Abscisic acid receptor PYL2/Protein phosphatase 2C 16
IC50: 10
1
2D 3D TSV 
Acetolactate synthase 2, chloroplastic
IC50: 12
1
2D 3D TSV 
Acetolactate synthase catalytic subunit, mitochondrial
Ki: 8 IC50: 1
2
2D 3D TSV 
Acetylcholine receptor subunit alpha/Neuronal acetylcholine receptor subunit beta-2
Ki: 8 EC50: 1
4
2D 3D TSV 
Acidic phospholipase A2 CM-I
Ki: 9
1
2D 3D TSV 
Acyl-[acyl-carrier-protein]--UDP-N-acetylglucosamine O-acyltransferase
IC50: 1 Kd: 8
2
2D 3D TSV 
Adenylate cyclase type 4
Ki: 9
1
2D 3D TSV 
ALK tyrosine kinase receptor [C1156Y]
IC50: 10
2
2D 3D TSV 
Alpha-1-antitrypsin-related protein
IC50: 9
1
2D 3D TSV 
Alpha-tocopherol transfer protein
Kd: 9
1
2D 3D TSV 
Anthranilate--CoA ligase
Ki: 9
2
2D 3D TSV 
ATP synthase subunit beta, mitochondrial
IC50: 9
1
2D 3D TSV 
Beta-N-acetylhexosaminidase
Ki: 9
2
2D 3D TSV 
Breakpoint cluster region protein
IC50: 9
1
2D 3D TSV 
Bromodomain-containing protein 2 [348-455]
Ki: 2 Kd: 8
2
2D 3D TSV 
CAD protein
Ki: 6 IC50: 4
3
2D 3D TSV 
Camphor 5-monooxygenase
IC50: 9
1
2D 3D TSV 
Carnitine monooxygenase oxygenase/reductase subunit
IC50: 9
1
2D 3D TSV 
Carnitine palmitoyl transferase I liver isoform
IC50: 9
1
2D 3D TSV 
Cell division related protein kinase 2
IC50: 9
1
2D 3D TSV 
Coagulation factor V
IC50: 23
1
2D 3D TSV 
Cytochrome P450 2D1
IC50: 9
1
2D 3D TSV 
Cytosolic endo-beta-N-acetylglucosaminidase
Ki: 2 IC50: 10
5
2D 3D TSV 
Diacylglycerol kinase zeta
IC50: 22
3
2D 3D TSV 
Dihydrofolate reductase type 1 from Tn4003
IC50: 9
1
2D 3D TSV 
DNA ligase A
IC50: 13
3
2D 3D TSV 
DNA-directed DNA polymerase
IC50: 9
3
2D 3D TSV 
DNA-directed DNA/RNA polymerase mu
IC50: 9
3
2D 3D TSV 
Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1
Ki: 8
1
2D 3D TSV 
Dual specificity protein phosphatase 10
Ki: 4 IC50: 6
6
2D 3D TSV 
Dual specificity tyrosine-phosphorylation-regulated kinase 4
IC50: 11
9
2D 3D TSV 
EH domain-containing protein 1
IC50: 8 Kd: 3
1
2D 3D TSV 
Elongin-B/Elongin-C/Hypoxia-inducible factor 1-alpha/von Hippel-Lindau disease tumor suppressor
IC50: 9
1
2D 3D TSV 
Eosinophil peroxidase
IC50: 9
3
2D 3D TSV 
Epidermal growth factor receptor [696-1022,L858R]
IC50: 7 Kd: 4
3
2D 3D TSV 
Fibroblast growth factor 23
IC50: 9
1
2D 3D TSV 
GABA(A) receptor-associated protein
Ki: 10
1
2D 3D TSV 
Gag-Pol polyprotein [484-582,I497V,V499I,E519D,G532V,I538V,R541K,D544E,Q553K,V566A,L573M]
Ki: 9
1
2D 3D TSV 
Gag-Pol polyprotein [588-1027,K691N]/[588-1147,K690N]
Ki: 5 IC50: 5
2
2D 3D TSV 
Gag-Pol polyprotein [600-1027,G789A]/[600-1155,G789A]
IC50: 9
2
2D 3D TSV 
Gag-Pol polyprotein [600-1027,V705A]/[600-1155,V705A]
IC50: 9
2
2D 3D TSV 
Gag-Pol polyprotein [600-1028,C879S]/[600-1151,C879S]
IC50: 18
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-4/beta-2/gamma-2
EC50: 18
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit rho-2
IC50: 3 Kd: 1 EC50: 6
2
2D 3D TSV 
Glutamate receptor ionotropic, kainate 4
Ki: 11
2
2D 3D TSV 
Guanine nucleotide-binding protein subunit alpha-11
IC50: 15
1
2D 3D TSV 
Histone deacetylase 6 [440-798]
Ki: 8 IC50: 8 Kd: 1
1
2D 3D TSV 
Histone-lysine N-methyltransferase, H3 lysine-79 specific [1-416]
IC50: 9
1
2D 3D TSV 
HIV-1 Protease Mutant (L10I/L90M)
ITC: 9
2
0
2D 3D TSV 
HIV-1 Protease Mutant (M46I/I54V)
ITC: 9
2
0
2D 3D TSV 
HIV-1 Protease Mutant (V82A/I84V)
ITC: 9
2
0
2D 3D TSV 
HIV-1 Protease Mutant, MDR-HM
ITC: 9
2
0
2D 3D TSV 
HIV-1 Protease Mutant, MDR-QM
ITC: 9
2
0
2D 3D TSV 
Interleukin-22 receptor subunit alpha-2
IC50: 9
1
2D 3D TSV 
Isoform PNNOS of Nitric oxide synthase, brain (PNNOS) -973,I269V,M336V,D597N]
Ki: 5 Kd: 4
2
2D 3D TSV 
Kinase suppressor of Ras 2
IC50: 10
3
2D 3D TSV 
LIP1, secretory lipase (Family 3)
IC50: 11
1
2D 3D TSV 
Lysine-specific demethylase 5A [1-739]
IC50: 9
1
2D 3D TSV 
Meprin A subunit alpha
IC50: 10
2
2D 3D TSV 
Monocarboxylate transporter 2
Ki: 5 IC50: 4
1
2D 3D TSV 
Myc proto-oncogene protein/Protein max
IC50: 15 Kd: 1
2
2D 3D TSV 
Neprilysin [1-24]
IC50: 9
1
2D 3D TSV 
Neuronal acetylcholine receptor subunit beta-4
Ki: 9
2
2D 3D TSV 
Oprd1b protein
Ki: 9
1
2D 3D TSV 
P2Y purinoceptor 13
EC50: 9
1
2D 3D TSV 
Penicillin-binding protein 2B
IC50: 76
3
2D 3D TSV 
Peptide-N(4)-(N-acetyl-beta-glucosaminyl)asparagine amidase
Kd: 9
1
2D 3D TSV 
Phenylalanine-4-hydroxylase
Ki: 9 IC50: 1
2
2D 3D TSV 
Phospholipase A1 member A
IC50: 10
1
2D 3D TSV 
Plasmepsin IV, putative
Ki: 10
1
2D 3D TSV 
Polycystin-1
Ki: 12
1
2D 3D TSV 
Polynucleotide kinase
IC50: 9
3
2D 3D TSV 
Primary amine oxidase
IC50: 9
1
2D 3D TSV 
Pro-neuropeptide Y
Ki: 13
4
2D 3D TSV 
Proto-oncogene tyrosine-protein kinase Src [251-533,T338M]
IC50: 6 Other: 3
1
2D 3D TSV 
Pyrazinamidase/nicotinamidase, PncA protein
Ki: 9
1
2D 3D TSV 
Pyruvate dehydrogenase E1 component subunit beta, mitochondrial
IC50: 10
2
2D 3D TSV 
Rat vasopressin-neurophysin
Ki: 9
3
2D 3D TSV 
Rhizopuspepsin
Ki: 7 IC50: 2
3
2D 3D TSV 
Rhomboid protease GluP
IC50: 9
1
2D 3D TSV 
Ribonuclease H1
IC50: 9
3
2D 3D TSV 
Serine/threonine-protein kinase LMTK3
IC50: 9
1
2D 3D TSV 
Serine/threonine-protein kinase PIM
ITC: 9
1
2D 3D TSV 
Serine/threonine-protein kinase SIK3
IC50: 9 Kd: 1
5
2D 3D TSV 
Serine/threonine-protein kinase VRK1
IC50: 9 Kd: 1
6
2D 3D TSV 
Signal transducer and activator of transcription 1
Ki: 3 IC50: 6
4
2D 3D TSV 
Sodium- and chloride-dependent neutral and basic amino acid transporter B(0+)
IC50: 9
1
2D 3D TSV 
Somatostatin
Ki: 9
8
2D 3D TSV 
Splicing factor 45
Kd: 9
1
2D 3D TSV 
Transcription factor ETV6/Vascular endothelial growth factor receptor 2
IC50: 9
1
2D 3D TSV 
Trehalose-phosphatase
Ki: 9
1
2D 3D TSV 
Tumor necrosis factor ligand superfamily member 10
IC50: 20
2
2D 3D TSV 
Tyrosine-protein kinase ABL1 [Y253F]
Ki: 10
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 8
IC50: 9
5
2D 3D TSV 
UDP-glucuronosyltransferase 1A9
Ki: 6 IC50: 3
7
2D 3D TSV 
Vitamin D3 receptor A
Kd: 5 EC50: 8
3
2D 3D TSV