BDBM23183 5-(aminomethyl)-1,2-oxazol-3-ol::Agarin::CHEMBL273481::Muscimol::Pantherine
SMILES NCc1cc(=O)[nH]o1
InChI Key InChIKey=ZJQHPWUVQPJPQT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 28 hits for monomerid = 23183
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-5(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-6(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-3(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-1(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit alpha-2(Homo sapiens (Human))
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp and Dohme Research Laboratories
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid type B receptor subunit 1(Rattus norvegicus (Rat))
TBA
Curated by PDSP Ki Database
TBA
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit rho-3(Homo sapiens (Human))
University of Alabama At Birmingham
Curated by PDSP Ki Database
University of Alabama At Birmingham
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
TargetGamma-aminobutyric acid receptor subunit rho-2(Homo sapiens (Human))
University Of Sydney
Curated by ChEMBL
University Of Sydney
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Partial agonist activity against human rho-2 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Agonist activity at human GABAA rho1 receptor expressed in TSA201 cells after 1 min by FLIPR assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Partial agonist activity at GABAC rho1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKd: 2.30E+3nMAssay Description:Partial agonist activity against human rho-1 subunit GABA-C receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:In vitro inhibition of [3H]-GABA binding to Gamma-aminobutyric-acid receptor of rat brain synaptic membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMpH: 8.5 T: 2°CAssay Description:D-amino acid oxidase (DAAO) was assayed in a 96-well plate format. D-serine was oxidatively deaminated by porcine D-amino acid oxidase in the presenc...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1/GABA transporter 2/GABA transporter 3/betaine transporter(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 3.20E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit rho-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clamp m...More data for this Ligand-Target Pair