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BDBM10846 4-(1H-indol-2-yl)pyrimidin-2-amine::isomeridianin G

SMILES: Nc1nccc(n1)-c1cc2ccccc2[nH]1

InChI Key: InChIKey=DMIMDIGPBYDVRA-UHFFFAOYSA-N

Data: 6 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 10846
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1 (Human)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.40E+5	n/a	n/a	n/a	n/a	7.2	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-dependent kinase 5 activator 1 [99-307] (Human)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.30E+5	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
cAMP-dependent protein kinase catalytic subunit alpha (Bovine)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	5.00E+5	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
cGMP-dependent protein kinase 1 (Bovine)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.00E+6	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glycogen synthase kinase-3 beta (Rat)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	4.20E+5	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Glycogen synthase kinase-3 beta (Human)	BDBM10846 (4-(1H-indol-2-yl)pyrimidin-2-amine \| isomeridianin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	4.20E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair