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BDBM12024 4-Arylazo-3,5-diamino-1H-pyrazole 1b::4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamine

SMILES: Nc1n[nH]c(N)c1\N=N\c1ccccc1

InChI Key: InChIKey=BLXRKDXUWQFGAW-UHFFFAOYSA-N

Data: 6 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 12024
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.2	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-dependent kinase 2/G1/S-specific cyclin-E1 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.00E+5	n/a	n/a	n/a	n/a	7.2	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-dependent kinase 4/G1/S-specific cyclin-D1 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	7.2	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-H/Cyclin-dependent kinase 7 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-T1/Cyclin-dependent kinase 9 (Human)	BDBM12024 (4-[(E)-2-phenyldiazen-1-yl]-1H-pyrazole-3,5-diamin...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.50E+4	n/a	n/a	n/a	n/a	n/a	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair