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BDBM193117 US10526329, Compound 192::US11072611, Compound 192::US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)piperazin-1-yl)-2-ethylimidazo[1,2-a]pyridin-3-yl)-4-(4-fluorophenyl)-N-methylthiazol-2-amine

SMILES: CCc1nc2ccc(cn2c1N(C)c1nc(cs1)-c1ccc(F)cc1)N1CCN(Cc2cnc[nH]2)CC1

InChI Key: InChIKey=REMDJYSRAUFISE-UHFFFAOYSA-N

Data: 7 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 193117   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 750n/an/an/an/a8.525


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 750n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 50n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 750n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 50n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Rat)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 4.10E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Autotaxin


(Human)
BDBM193117
PNG
(US9670204, 192 N-(6-(4-((1H-imidazol-5-yl)methyl)p...)
GoogleScholar
UniChem
n/an/a 771n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair