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BDBM201222 US9233968, 25

SMILES: O=C(Nc1cccc(c1)C#Cc1ccc2nccn2n1)c1cc2ccccc2o1

InChI Key: InChIKey=GXCSUVBPKJBUPR-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 201222
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Vascular endothelial growth factor receptor 2 (Human)	BDBM201222 (US9233968, 25) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.61E+3	n/a	n/a	n/a	n/a	7.4	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Human)	BDBM201222 (US9233968, 25) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.72E+3	n/a	n/a	n/a	n/a	7.4	30
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM201222 (US9233968, 25) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor beta (Human)	BDBM201222 (US9233968, 25) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	37
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair