BDBM225248 4-(tert-Butyl)-N-(2-phenylbenzo[d]oxazol-6-yl)benzenesulfonamide (9)

SMILES CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc1ccc2nc(oc2c1)-c1ccccc1

InChI Key InChIKey=DFUZLOZWENCKSN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 225248   

TargetHistone-lysine N-methyltransferase EHMT2(Human)
Shenyang Pharmaceutical University

LigandPNGBDBM225248(4-(tert-Butyl)-N-(2-phenylbenzo[d]oxazol-6-yl)benz...)
Affinity DataIC50: 3.63E+4nMpH: 8.5 T: 2°CAssay Description:Biochemical activity of G9a was measured as described [Kubicek et al., Mol. Cell, 25:473-481]. Assays were performed in white, opaque 384-well plates...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed