BDBM23028 (9Z)-octadec-9-enamide::14C-labeled oleamide::CHEMBL15927::Oleamide::Oleic acid amide::Oleylamide

SMILES CCCCCCCC\C=C/CCCCCCCC(N)=O

InChI Key InChIKey=FATBGEAMYMYZAF-KTKRTIGZSA-N

Data  1 KI  6 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 23028   

TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£ Catholique de Louvain

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibition of [3H]CP-55940 binding to rat cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Rattus norvegicus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universit£ Catholique de Louvain

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of fatty acid amide hydrolase; range = 22-68 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rattus norvegicus)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | 14C-labeled oleamide | CH...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed