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BDBM238524 US9394297, 156::US9394297, 160::US9394297, 161

SMILES: CC1CNC(=O)c2cc([nH]c12)-c1cccc2nc(C)c(F)nc12

InChI Key: InChIKey=UAYKLVYFPJYTBE-UHFFFAOYSA-N

Data: 6 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 238524
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Serine/threonine-protein kinase pim-1 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	526	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-1 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.800	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	758	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.5	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Serine/threonine-protein kinase pim-2 (Human)	BDBM238524 (US9394297, 161 \| US9394297, 160 \| US9394297, 156) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.700	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair