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BDBM259526 US9505749, 37

SMILES: Cc1cc(=O)[nH]c(SCCC(=O)N[C@H]2CC[C@@H](CC2)c2nnc(o2)-c2ccccc2)n1

InChI Key: InChIKey=ZFHIMDPSSCABJV-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 259526
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Poly [ADP-ribose] polymerase 1 (Human)	BDBM259526 (US9505749, 37) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>8.50E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Poly [ADP-ribose] polymerase tankyrase-1 [1091-1325] (Human)	BDBM259526 (US9505749, 37) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.70	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Poly [ADP-ribose] polymerase tankyrase-2 [946-1162] (Human)	BDBM259526 (US9505749, 37) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.48	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Poly [ADP-ribose] polymerase 2 (Human)	BDBM259526 (US9505749, 37) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.70E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair