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BDBM27077 N-[3-(1H-1,3-benzodiazol-2-yl)-1H-pyrazol-4-yl]acetamide::pyrazole-benzimidazole amide analogue, 6

SMILES: CC(=O)Nc1c[nH]nc1-c1nc2ccccc2[nH]1

InChI Key: InChIKey=LEFKZSWCBZBDLU-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 27077
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Aurora kinase A (Human)	BDBM27077 (N-[3-(1H-1,3-benzodiazol-2-yl)-1H-pyrazol-4-yl]ace...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	70	n/a	n/a	n/a	n/a	7.0	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Aurora kinase B (Human)	BDBM27077 (N-[3-(1H-1,3-benzodiazol-2-yl)-1H-pyrazol-4-yl]ace...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	510	n/a	n/a	n/a	n/a	8.5	22
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1 (Human)	BDBM27077 (N-[3-(1H-1,3-benzodiazol-2-yl)-1H-pyrazol-4-yl]ace...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	3.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM27077 (N-[3-(1H-1,3-benzodiazol-2-yl)-1H-pyrazol-4-yl]ace...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	990	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair