BDBM277782 N-cyano-3-({5-chloro-1-[2-(pyrrolidin-1-yl)ethyl]-1H-indazol-3-yl}amino)pyridine-4-carboxamide, formic acid salt::US10040779, Example 79::US10336727, Example 79::US9617242, Example 79Biochemical

SMILES: Clc1ccc2n(CCN3CCCC3)nc(Nc3cnccc3C(=O)NC#N)c2c1

InChI Key: InChIKey=COKQEBSDGZNRLI-UHFFFAOYSA-N

Data: 3 IC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 277782   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Lysine-specific demethylase 5A (Human)	BDBM277782 (N-cyano-3-({5-chloro-1-[2-(pyrrolidin-1-yl)ethyl]-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
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Lysine-specific demethylase 5B (Human)	BDBM277782 (N-cyano-3-({5-chloro-1-[2-(pyrrolidin-1-yl)ethyl]-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	<100	n/a	n/a	n/a	n/a	n/a	n/a
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					More data for this Ligand-Target Pair
Lysine-specific demethylase 4C (Human)	BDBM277782 (N-cyano-3-({5-chloro-1-[2-(pyrrolidin-1-yl)ethyl]-...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	550	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
					More data for this Ligand-Target Pair