BDBM29083 Impulsin::MimyX::Palmidrol::Palmityoletanolamide (PEA)

SMILES CCCCCCCCCCCCCCCC(=O)NCCO

InChI Key InChIKey=HXYVTAGFYLMHSO-UHFFFAOYSA-N

Data  2 KI  3 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 29083   

TargetCannabinoid receptor 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataKi: >5.00E+3nM ΔG°: >-7.35kcal/molepH: 7.4 T: 30°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataKi: >5.00E+3nM ΔG°: >-7.35kcal/molepH: 7.4 T: 30°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rat)
Ghent University

Curated by ChEMBL
LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of rat recombinant FAAH assessed as [3H]AEA hydrolysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
Universita Del Piemonte Orientale

LigandPNGBDBM29083(Impulsin | MimyX | Palmidrol | Palmityoletanolamid...)
Affinity DataEC50: >1.00E+4nMAssay Description:The effect of the substances on Ca2+ influx was determined by using HEK-293 cells stably overexpressing recombinant human TRPV1 cDNA. The cells were ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed