BDBM292474 (R)-(2-(aminomethyl)piperidin-1-yl)(2-(tert-butyl)-6-(5-phenylpyrazolo[1,5-a]pyrimidin-3-yl)pyridin-4-yl)methanone::US10100058, Example 130

SMILES CC(C)(C)c1cc(cc(n1)-c1cnn2ccc(nc12)-c1ccccc1)C(=O)N1CCCC[C@@H]1CN

InChI Key InChIKey=AGRPDXNCSXDDCP-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 292474   

LigandChemical structure of BindingDB Monomer ID 292474BDBM292474(US10100058, Example 130 | (R)-(2-(aminomethyl)pipe...)
Affinity DataIC50: 266nMAssay Description:The biochemical activity of recombinant CaMKIIδ was measured by monitoring the phosphorylation of a target peptide using Homogenous Time Resolve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2019
Entry Details
US Patent