BDBM31889 BMS 961::BMS270394::BMS961
SMILES CC1(C)CCC(C)(C)c2cc(ccc12)[C@@H](O)C(=O)Nc1ccc(cc1F)C(O)=O
InChI Key InChIKey=AANFHDFOMFRLLR-LJQANCHMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 31889
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 1.5nM ΔG°: -11.2kcal/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKd: 528nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair