BDBM434384 US10562891, Example 303::US11008308, Example 303
SMILES F[C@@H]1CNCC[C@@H]1SCc1nc2cc(NCC3CCC3)c(F)cc2c(=O)[nH]1
InChI Key
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 434384
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP14 [1611-1801](Homo sapiens (Human))
Ribon Therapeutics
US Patent
Ribon Therapeutics
US Patent
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair