BDBM434510 US10562891, Example 424::US11008308, Example 424

SMILES COCC(=O)N1CCC(COc2cc(F)c3c(c2)nc(CSC2CCOCC2)[nH]c3=O)CC1

InChI Key InChIKey=PEVYFKITQYTFNT-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 434510   

TargetProtein mono-ADP-ribosyltransferase PARP14(Homo sapiens (Human))
Ribon Therapeutics

US Patent
LigandPNGBDBM434510(US10562891, Example 424 | US11008308, Example 424)
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProtein mono-ADP-ribosyltransferase PARP14 [1611-1801](Homo sapiens (Human))
Ribon Therapeutics

US Patent
LigandPNGBDBM434510(US10562891, Example 424 | US11008308, Example 424)
Affinity DataIC50: <1.00E+3nMAssay Description:Enzymatic inhibition of PARP14 was measured using a dissociation-enhanced lanthanide fluorescence immunoassay (DELFIA) monitoring the auto-modificati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent