BDBM499486 US11020395, Example 16.0::US11046680, Example 329.0::US11191762, Example 48.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)N\C(S)=N/c1c(OC)cccc1OC)c1ncc(C)cn1

InChI Key InChIKey=CHHPSMFZWCGLIQ-LRDDRELGSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 499486   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM499486(US11020395, Example 16.0 | US11046680, Example 329...)
Affinity DataEC50:  22nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM499486(US11020395, Example 16.0 | US11046680, Example 329...)
Affinity DataEC50:  440nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM499486(US11020395, Example 16.0 | US11046680, Example 329...)
Affinity DataEC50:  0.200nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent