BDBM499617 US11020395, Example 217.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc(n1-c1c(OC)cccc1OC)C12CC(C1)C2)c1ncc(Cl)cn1

InChI Key InChIKey=VGTVHXSNZNPQGR-JAVUXCMTSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 499617   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM499617(US11020395, Example 217.0)
Affinity DataEC50:  7.40nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent