BDBM50010052 2-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl]-2H-naphtho[1,8-cd]isothiazole 1,1-dioxide::CHEMBL440134
SMILES O=S1(=O)N(CCCCN2CCC(=CC2)c2ccccc2)c2cccc3cccc1c23
InChI Key InChIKey=OKJRBFNMYSRTKZ-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50010052
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
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Curated by ChEMBL
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer
Curated by ChEMBL
Affinity DataIC50: 7.80nMAssay Description:The concentration required to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat brain membranes was measured (in vitro)More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(RAT)
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Curated by ChEMBL
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:The concentration required to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat brain membranes (in vitro)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
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Curated by ChEMBL
Centre De Recherches De Vitry Alfortville Rh£Ne-Poulenc Rorer
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:The concentration required to inhibit [3H]spiperone binding to dopamine receptor D2 in rat brain membranes (in vitro)More data for this Ligand-Target Pair