BDBM50026994 CHEMBL2113646
SMILES [H][C@@]12Oc3c4c(C[C@@]5([H])N(CC6CC6)CC[C@@]14[C@]5(Cc1c2oc2ccccc12)OCC)ccc3O
InChI Key InChIKey=WGBLEWOROOAZNK-CSZVXOJQSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50026994
Affinity DataKi: 0.880nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by DAMGO (Opioid receptor mu 1) antagonistMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by U69,593 (Opioid receptor kappa 1) antagonistMore data for this Ligand-Target Pair