BDBM50027284 2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-phenyl}-1H-benzoimidazole-5-carboxamidine::CHEMBL101672

SMILES NC(=N)c1ccc(OCCCCCOc2ccc(cc2)-c2nc3ccc(cc3[nH]2)C(N)=N)cc1

InChI Key InChIKey=HRVAWGMMOAKYTG-UHFFFAOYSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50027284   

TargetSerine protease 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  1.44E+3nMAssay Description:Inhibition constant against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  2.24E+3nMAssay Description:Inhibition constant against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  2.24E+3nMAssay Description:Competitive reversible inhibition of bovine thrombin using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after 15 to 40 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  3.83E+3nMAssay Description:Inhibition constant against human plasminogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlandular kallikrein(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  5.16E+3nMAssay Description:Competitive reversible inhibition of porcine pancreatic kallikrein using alpha-N-benzoyl-DL-arginine-p-nitroanilide hydrochloride as substrate after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50027284(2-{4-[5-(4-Carbamimidoyl-phenoxy)-pentyloxy]-pheny...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition constant against UrokinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed