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BDBM50071714 1-[4-(8-Chloro-10-methyl-10,11-dihydro-5H-4,10-diaza-dibenzo[a,d]cyclohepten-5-yl)-piperazin-1-yl]-2-pyridin-4-yl-ethanone::CHEMBL82505
SMILES: CN1Cc2cccnc2C(N2CCN(CC2)C(=O)Cc2ccncc2)c2ccc(Cl)cc12
InChI Key: InChIKey=UPAXVBQVDHBZJD-UHFFFAOYSA-N
Data: 1 IC50
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha (Human) | BDBM50071714![]() (1-[4-(8-Chloro-10-methyl-10,11-dihydro-5H-4,10-dia...) | GoogleScholar | UniChem | n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||