BDBM50119392 CHEMBL141845::N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)H-pyrazolo[1,5-a]pyridine-3-carboxamide::Pyrazolo[1,5-a]pyridine-3-carboxylic acid {2-[4-(2-methoxy-phenyl)-piperazin-1-yl]-ethyl}-amide

SMILES COc1ccccc1N1CCN(CCNC(=O)c2cnn3ccccc23)CC1

InChI Key InChIKey=XJGIQRQUJHWFSC-UHFFFAOYSA-N

Data  10 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50119392   

TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  0.670nMAssay Description:Biniding affinity for Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  0.670nMAssay Description:Binding affinity for human Dopamine receptor D4 by [3H]- spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cell membranes by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  140nMAssay Description:Binding affinity for human Dopamine receptor D2 (short) by [3H]- spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  290nMAssay Description:Binding affinity for human dopamine receptor D2 longMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  290nMAssay Description:Binding affinity for human Dopamine receptor D2 (long) by [3H]- spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  360nMAssay Description:Binding affinity for human dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  360nMAssay Description:Binding affinity for human Dopamine receptor D3 by [3H]- spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]ketanserin from human 5-HT2A receptor expressed in HEK293 cell membranes by radioligand competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander University

Curated by ChEMBL
LigandPNGBDBM50119392(CHEMBL141845 | N-(2-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity for porcine Dopamine receptor D1 by [3H]-SCH- 23390 displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed