BDBM50125886 2-Amino-N-{(R)-1-[(R)-1-formylamino-2-(1H-indol-3-yl)-ethylcarbamoyl]-2-1H-indol-3-yl-ethyl}-2-methyl-propionamide::AEZS-130::ARD-07::CHEMBL278623::EP-1572::JMV-1843::Macimorelin::Macimorelin acetate::aminoisobutyryl-tryptophyl-tryptophanamine-formyl

SMILES CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](Cc1c[nH]c2ccccc12)NC=O

InChI Key InChIKey=UJVDJAPJQWZRFR-DHIUTWEWSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50125886   

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50125886(2-Amino-N-{(R)-1-[(R)-1-formylamino-2-(1H-indol-3-...)
Affinity DataIC50:  22.9nMAssay Description:Binding affinity towards human pituitary Growth hormone secretagogue receptor using [125I][Tyr4]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50125886(2-Amino-N-{(R)-1-[(R)-1-formylamino-2-(1H-indol-3-...)
Affinity DataIC50:  123nMAssay Description:Binding affinity towards cloned human Growth hormone secretagogue receptor type I in LLC PK-1 cells using [125I][His9]-ghrelin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed