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BDBM50142024 3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-pyrrolo[2,3-b]pyridin-2-one::CHEMBL172179

SMILES: Cn1cc(\C=C2/C(=O)Nc3ncccc23)c2ccccc12

InChI Key: InChIKey=RJBBKRZRJMHITR-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50142024
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
High affinity nerve growth factor receptor (Human)	BDBM50142024 (3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-py...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2 (Human)	BDBM50142024 (3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-py...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>6.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
RAF proto-oncogene serine/threonine-protein kinase (Human)	BDBM50142024 (3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-py...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	7.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
High affinity nerve growth factor receptor (Human)	BDBM50142024 (3-(1-Methyl-1H-indol-3-ylmethylene)-1,3-dihydro-py...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair