BDBM501842 4-{1-methyl-5-[4- (methylamino)piperidyl]-2-(4- methylphenyl)-6-oxo-3- hydropyridyl}benzenecarbonitrile::US11028066, Example 80
SMILES CNC1CCN(CC1)c1cc(-c2ccc(cc2)C#N)c(-c2ccc(C)cc2)n(C)c1=O
InChI Key InChIKey=TYZJQHVYGBCYAK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 501842
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Celgene Quanticel Research
US Patent
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of LSD1 activity is based on Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The inhibitory properties ...More data for this Ligand-Target Pair