BDBM501931 US11028075, Example 64
SMILES Fc1cc(O[C@H]2CC[C@@H](C[C@@H]2N2CCCC2)c2cccc(OC(F)(F)F)c2)c(Cl)cc1S(=O)(=O)Nc1ccncn1
InChI Key InChIKey=DFHGNSWUHXYPHU-TZYHBYERSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 501931
Affinity DataIC50: 0.554nMAssay Description:The following voltage clamp electrophysiology studies are performed on representative compounds using cells heterologously expressing Nav1.7 or Nav1....More data for this Ligand-Target Pair
Affinity DataIC50: 1.37nMAssay Description:Saturation experiments. A competitive NaV1.7 inhibitor having a methyl group is tritiated. Three tritiums are incorporated in place of methyl hydroge...More data for this Ligand-Target Pair