BDBM50198795 7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylpiperazin-1-yl)ethoxy)phenyl)benzo[e][1,2,4]triazin-3-amine::CHEMBL230615::US8481536, 379::US8481536, 580

SMILES CN1CCN(CCOc2cccc(Nc3nnc4cc(cc(C)c4n3)-c3c(C)cccc3C)c2)CC1

InChI Key InChIKey=LARRSIBKNUNYRQ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50198795   

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50198795(7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylp...)
Affinity DataIC50:  39.5nMT: 2°CAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50198795(7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylp...)
Affinity DataIC50:  40nMAssay Description:Inhibition of SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Targegen

US Patent
LigandPNGBDBM50198795(7-(2,6-dimethylphenyl)-5-methyl-N-(3-(2-(4-methylp...)
Affinity DataIC50:  69.1nMAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair
In DepthDetails US Patent