BDBM50200028 2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)-benzamide::CHEMBL376092

SMILES COc1ccccc1C1CCN(CNC(=O)c2cccc(C)c2)CC1

InChI Key InChIKey=LAFUMJMKVVCEGP-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50200028   

TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50200028(2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipy...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]A369508 from human D4 receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50200028(2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipy...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]7-OH-PIPAT from human D2L receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50200028(2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipy...)
Affinity DataEC50:  206nMAssay Description:Agonist activity at human D4.4 receptor in HEK293 cells coexpressing Galphaqo5 by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50200028(2-methoxy-N-(3',4',5',6'-tetrahydro-2'H-[2,4'-bipy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human D2 receptor in HEK293 cells coexpressing Galphaqo5 by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed