BDBM50232355 (3aR,6aR)-2-(cyclopropylmethyl)-6-(4-(2-(pyrrolidin-1-yl)ethyl)phenyl)-1,2,3,3a,4,6a-hexahydrocyclopenta[c]pyrrole::CHEMBL408934
SMILES C(Cc1ccc(cc1)C1=CC[C@H]2CN(CC3CC3)C[C@@H]12)N1CCCC1
InChI Key InChIKey=SMDURVDNVKUIAT-JTHBVZDNSA-N
Data 5 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50232355
Affinity DataKi: 0.0700nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortex membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of N-[3H]methylhistamine from histamine H3 receptor in rat cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Antagonist activity at human histamine H3 receptor expressed in CHOK1 cells by [3H]R(-)-alpha-methylhistamine displacement assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inverse agonist activity at human H3 receptor expressed in CHOK1 cells by GTPgammaS binding assayMore data for this Ligand-Target Pair