BDBM50243347 CHEMBL4064244

SMILES Oc1ccc(\C=C\c2cc(Br)c(O)c(Br)c2)cc1

InChI Key InChIKey=KGDYRCIWRHRFPK-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50243347   

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50243347(CHEMBL4064244)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TRPA1 expressed in HEK293 cells assessed as induction of calcium influx at 30 uM after 6 mins by Fluo-4 dye-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hyogo University of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50243347(CHEMBL4064244)
Affinity DataIC50: 1.61E+4nMAssay Description:Inhibition of human TRPA1 expressed in HEK293 cells assessed as decrease in AITC-induced calcium influx preincubated for 6 mins followed by AITC addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed