BDBM50257340 CHEMBL4072828

SMILES: FC(F)(F)c1ccccc1CNC(=O)c1cccc(NCc2nnc3-c4ccncc4OCCn23)c1

InChI Key: InChIKey=DMNINFHJFPFPIZ-UHFFFAOYSA-N

Data: 7 IC50  1 EC50

Find this compound or compounds like it in BindingDB or PDB:

Substructure Similarity at least:  must be >=0.5 Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50257340   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Rhodopsin kinase GRK1 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	270	n/a	n/a	n/a	n/a	n/a	n/a
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G protein-coupled receptor kinase 5 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
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G protein-coupled receptor kinase 6 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>3.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
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Beta-adrenergic receptor kinase 2 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	0.650	n/a	n/a	n/a	n/a	n/a	n/a
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Rhodopsin kinase GRK7 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	2.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
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Beta-adrenergic receptor kinase 1 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	n/a	n/a	1.50E+3	n/a	n/a	n/a	n/a
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Beta-adrenergic receptor kinase 1 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
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Rho-associated protein kinase 2 (Human)	BDBM50257340 (CHEMBL4072828) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	49	n/a	n/a	n/a	n/a	n/a	n/a
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