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BDBM50260889 3-(2-aminoquinazolin-6-yl)-4-methyl-1-phenylpyridin-2(1H)-one::CHEMBL523741

SMILES: Cc1ccn(-c2ccccc2)c(=O)c1-c1ccc2nc(N)ncc2c1

InChI Key: InChIKey=LHHCZOUDWJLWHD-UHFFFAOYSA-N

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50260889
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mast/stem cell growth factor receptor Kit (Human)	BDBM50260889 (3-(2-aminoquinazolin-6-yl)-4-methyl-1-phenylpyridi...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	210	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Human)	BDBM50260889 (3-(2-aminoquinazolin-6-yl)-4-methyl-1-phenylpyridi...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Tyrosine-protein kinase Lck (Human)	BDBM50260889 (3-(2-aminoquinazolin-6-yl)-4-methyl-1-phenylpyridi...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
Proto-oncogene tyrosine-protein kinase Src (Human)	BDBM50260889 (3-(2-aminoquinazolin-6-yl)-4-methyl-1-phenylpyridi...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	990	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair