BDBM50277340 1-methyl-N-(4-methyl-3-(morpholinosulfonyl)phenyl)cyclohexanecarboxamide::CHEMBL515866

SMILES Cc1ccc(NC(=O)C2(C)CCCCC2)cc1S(=O)(=O)N1CCOCC1

InChI Key InChIKey=KLRDRQKZOQEROV-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50277340   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277340(1-methyl-N-(4-methyl-3-(morpholinosulfonyl)phenyl)...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]CP55940 from human cloned CB2 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277340(1-methyl-N-(4-methyl-3-(morpholinosulfonyl)phenyl)...)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]CP55940 from human cloned CB1 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277340(1-methyl-N-(4-methyl-3-(morpholinosulfonyl)phenyl)...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human cloned CB2 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed