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BDBM50284089 CHEMBL355149::Pyrazolo[1,5-a]pyridine-3-carboxylic acid (8-methyl-8-aza-bicyclo[3.2.1]oct-3-yl)-amide

SMILES: CN1C2CCC1CC(C2)NC(=O)c1cnn2ccccc12

InChI Key:

Data: 4 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50284089
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
5-hydroxytryptamine receptor 3A/3B (Rat)	BDBM50284089 (Pyrazolo[1,5-a]pyridine-3-carboxylic acid (8-methy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	34	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 1A (Human)	BDBM50284089 (Pyrazolo[1,5-a]pyridine-3-carboxylic acid (8-methy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
D(2) dopamine receptor (Human)	BDBM50284089 (Pyrazolo[1,5-a]pyridine-3-carboxylic acid (8-methy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair
5-hydroxytryptamine receptor 3A/3B (Rat)	BDBM50284089 (Pyrazolo[1,5-a]pyridine-3-carboxylic acid (8-methy...) Show SMILES Show InChI	GoogleScholar	UniChem		n/a	n/a	105	n/a	n/a	n/a	n/a	n/a	n/a
TBA									Citation and Details
TBA					More data for this Ligand-Target Pair