BindingDB logo
myBDB logout

BDBM50329879 5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)pyridin-2(1H)-one::CHEMBL1271480

SMILES: O=c1ccc(c[nH]1)-c1cnn2cc(cnc12)-c1ccc(OCCN2CCOCC2)cc1

InChI Key: InChIKey=WMXDIPVFXWNELM-UHFFFAOYSA-N

Data: 7 IC50

Find this compound or compounds like it in BindingDB or PDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50329879   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Proto-oncogene tyrosine-protein kinase Src


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 61n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ephrin type-A receptor 2


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 260n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 1


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 470n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Vascular endothelial growth factor receptor 2


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 100n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Tyrosine-protein kinase Lck


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 430n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
MAP kinase-interacting serine/threonine-protein kinase 1


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 45n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair
Ribosomal protein S6 kinase alpha-1


(Human)
BDBM50329879
PNG
(5-(6-(4-(2-morpholinoethoxy)phenyl)pyrazolo[1,5-a]...)
GoogleScholar
UniChem
n/an/a 2.10E+3n/an/an/an/an/an/a


TBA



Citation and Details
More data for this
Ligand-Target Pair